Report error Found 63 Enz. Inhib. hit(s) with all data for entry = 50022547
Affinity DataIC50: 0.830nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged Plk1 (residues 1-603) expressed in baculovirus expression using casein as substrate in presence...More data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:Inhibition of recombinant human plk2 using casein as substrate in presence of gamma-[33P]-ATP by invitro kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged Plk3 (residues 19-301) using casein as substrate in presence of gamma-[33P]-ATP by invitro kin...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Affinity DataIC50: 2.41E+3nMAssay Description:Inhibition of PI3Ka (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 4.75E+3nMAssay Description:Inhibition of Met (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 6.55E+3nMAssay Description:Inhibition of Tie2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of HGFR (unknown origin)More data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-4(Human)
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Affinity DataIC50: 9.91E+3nMAssay Description:Inhibition of ErbB4 (unknown origin)More data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HER2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Hek (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GSK3beta (unknown origin)More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Flt3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of JAK3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of JAK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ITK (unknown origin)More data for this Ligand-Target Pair
TargetMAP kinase-activated protein kinase 2(Human)
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MAPKAP-K2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Lyn (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Lck (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of JNK1 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Human)
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MKK1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MSK1 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Human)
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MEK1 (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK1/cyclin B1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Btk (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Human)
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of B-RAF (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Beta IRK (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CK2 (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CK1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CHK1 (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ECK (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CSK (unknown origin)More data for this Ligand-Target Pair
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of C-RAF (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FGFR3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FGFR1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Src (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of SGK (unknown origin)More data for this Ligand-Target Pair
TargetMacrophage-stimulating protein receptor(Human)
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Ron (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ROCK2 (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 3(Human)
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR3 (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 1(Human)
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Syk (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of p38gamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of p38beta (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Nek6 (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Human)
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PDGFRb (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha(Human)
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Boehringer Ingelheim Austria GmbH
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PDGFRa (unknown origin)More data for this Ligand-Target Pair
