Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50019565
TargetMelanocyte-stimulating hormone receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205745((3S,6S,9R,12S,15S,23S)-15-[(2S)-2-aminohexanamido]...)
Affinity DataIC50: 0.200nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205745((3S,6S,9R,12S,15S,23S)-15-[(2S)-2-aminohexanamido]...)
Affinity DataEC50:  0.300nMAssay Description:Effect on human MC1R expressed in HEK293 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205745((3S,6S,9R,12S,15S,23S)-15-[(2S)-2-aminohexanamido]...)
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205745((3S,6S,9R,12S,15S,23S)-15-[(2S)-2-aminohexanamido]...)
Affinity DataIC50: 1.30nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205745((3S,6S,9R,12S,15S,23S)-15-[(2S)-2-aminohexanamido]...)
Affinity DataEC50:  1.90nMAssay Description:Effect on human MC3R expressed in HEK293 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205745((3S,6S,9R,12S,15S,23S)-15-[(2S)-2-aminohexanamido]...)
Affinity DataEC50:  2.90nMAssay Description:Effect on human MC4R expressed in HEK293 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205745((3S,6S,9R,12S,15S,23S)-15-[(2S)-2-aminohexanamido]...)
Affinity DataEC50:  3.30nMAssay Description:Effect on human MC5R expressed in HEK293 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205745((3S,6S,9R,12S,15S,23S)-15-[(2S)-2-aminohexanamido]...)
Affinity DataIC50: 7.5nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205746((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-5-(...)
Affinity DataIC50: 29nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205744((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-5-(...)
Affinity DataIC50: 43nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205743((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-2-b...)
Affinity DataIC50: 50nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205744((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-5-(...)
Affinity DataIC50: 87nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205746((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-5-(...)
Affinity DataIC50: 123nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205746((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-5-(...)
Affinity DataEC50:  180nMAssay Description:Effect on human MC5R expressed in HEK293 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205744((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-5-(...)
Affinity DataIC50: 580nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205746((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-5-(...)
Affinity DataEC50:  900nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205746((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-5-(...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205746((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-5-(...)
Affinity DataEC50: >1.00E+3nMAssay Description:Effect on human MC3R expressed in HEK293 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205744((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-5-(...)
Affinity DataIC50: 1.70E+3nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205746((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-5-(...)
Affinity DataIC50: 2.00E+3nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205744((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-5-(...)
Affinity DataEC50: >2.50E+3nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205743((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-2-b...)
Affinity DataIC50: 2.90E+3nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205746((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-5-(...)
Affinity DataEC50:  3.20E+3nMAssay Description:Effect on human MC4R expressed in HEK293 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205742((S)-3-((R)-2-acetamidohexanamido)-4-(2-((S)-1-((S)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205743((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-2-b...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human MC5R expressed in HEK293 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205743((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-2-b...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205743((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-2-b...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human MC4R expressed in HEK293 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205742((S)-3-((R)-2-acetamidohexanamido)-4-(2-((S)-1-((S)...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human MC4R expressed in HEK293 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205742((S)-3-((R)-2-acetamidohexanamido)-4-(2-((S)-1-((S)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205743((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-2-b...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human MC3R expressed in HEK293 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205743((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-2-b...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205742((S)-3-((R)-2-acetamidohexanamido)-4-(2-((S)-1-((S)...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human MC3R expressed in HEK293 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205742((S)-3-((R)-2-acetamidohexanamido)-4-(2-((S)-1-((S)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205742((S)-3-((R)-2-acetamidohexanamido)-4-(2-((S)-1-((S)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205744((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-5-(...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human MC5R expressed in HEK293 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205742((S)-3-((R)-2-acetamidohexanamido)-4-(2-((S)-1-((S)...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human MC5R expressed in HEK293 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205744((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-5-(...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human MC4R expressed in HEK293 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205742((S)-3-((R)-2-acetamidohexanamido)-4-(2-((S)-1-((S)...)
Affinity DataEC50: >1.00E+4nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205743((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-2-b...)
Affinity DataEC50: >1.00E+4nMAssay Description:Displacement of [125I]NDPalphaMSH from human MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50205744((2R,5S,8S,11S,19S)-19-[(2S)-2-aminohexanamido]-5-(...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human MC3R expressed in HEK293 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed