Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50019645
TargetLutropin-choriogonadotropic hormone receptor(Human)
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206401(N-((S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-y...)
Affinity DataKi:  0.311nMAssay Description:Displacement of [125I]hCG from LH receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLutropin-choriogonadotropic hormone receptor(Human)
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206401(N-((S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-y...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLutropin-choriogonadotropic hormone receptor(Human)
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206398(N-(4-hydroxyphenethyl)-5-(1-(4-tert-butylphenyl)-3...)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLutropin-choriogonadotropic hormone receptor(Human)
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206402(N-((S)-1-amino-3-(3-hydroxyphenyl)-1-oxopropan-2-y...)
Affinity DataEC50:  150nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLutropin-choriogonadotropic hormone receptor(Human)
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206399(N-((S)-2-amino-1-(4-hydroxyphenyl)-2-oxoethyl)-6-(...)
Affinity DataEC50:  170nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLutropin-choriogonadotropic hormone receptor(Human)
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206397((S)-N-(4-amino-4-oxo-1-phenylbutan-2-yl)-5-(1-(4-t...)
Affinity DataEC50:  190nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLutropin-choriogonadotropic hormone receptor(Human)
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206395((S)-N-(1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-y...)
Affinity DataEC50:  250nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLutropin-choriogonadotropic hormone receptor(Human)
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206400(N-((S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-y...)
Affinity DataEC50:  500nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLutropin-choriogonadotropic hormone receptor(Human)
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206405((S)-N-(1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-y...)
Affinity DataEC50:  2.30E+3nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLutropin-choriogonadotropic hormone receptor(Human)
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206403(N-((S)-1-amino-3-(4-tert-butoxyphenyl)-1-oxopropan...)
Affinity DataEC50:  1.21E+4nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLutropin-choriogonadotropic hormone receptor(Human)
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206396((S)-2-{3-[2-(4-tert-butyl-phenyl)-5-pyridin-3-yl-2...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLutropin-choriogonadotropic hormone receptor(Human)
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206404((S)-N-(1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-y...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed