Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50019645
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206401(CHEMBL246321 | N-((S)-1-amino-3-(4-hydroxyphenyl)-...)
Affinity DataKi:  0.311nMAssay Description:Displacement of [125I]-hCG from LH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206404((S)-N-(1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-y...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206400(CHEMBL247945 | N-((S)-1-amino-3-(4-hydroxyphenyl)-...)
Affinity DataEC50:  500nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206405((S)-N-(1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-y...)
Affinity DataEC50:  2.30E+3nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206401(CHEMBL246321 | N-((S)-1-amino-3-(4-hydroxyphenyl)-...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206397((S)-N-(4-amino-4-oxo-1-phenylbutan-2-yl)-5-(1-(4-t...)
Affinity DataEC50:  190nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206402(CHEMBL439392 | N-((S)-1-amino-3-(3-hydroxyphenyl)-...)
Affinity DataEC50:  150nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206399(CHEMBL247700 | N-((S)-2-amino-1-(4-hydroxyphenyl)-...)
Affinity DataEC50:  170nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206396((S)-2-{3-[2-(4-tert-butyl-phenyl)-5-pyridin-3-yl-2...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206395((S)-N-(1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-y...)
Affinity DataEC50:  250nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206403(CHEMBL269261 | N-((S)-1-amino-3-(4-tert-butoxyphen...)
Affinity DataEC50:  1.21E+4nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206398(CHEMBL429108 | N-(4-hydroxyphenethyl)-5-(1-(4-tert...)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed