Compile Data Set for Download or QSAR
Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 50019792
Target11-beta-hydroxysteroid dehydrogenase 1(Mouse)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207760([4-(2-hydroxy-ethyl)-piperazin-1-yl]-(3-p-tolyl-ad...)
Affinity DataIC50: 43nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO cells after 4 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207768(cid_2882437 | CHEMBL246338 | (4-methyl-piperazin-1...)
Affinity DataIC50: 80nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mouse)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207768(cid_2882437 | CHEMBL246338 | (4-methyl-piperazin-1...)
Affinity DataIC50: 81nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO cells after 4 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mouse)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207772(adamantan-1-yl-piperidin-1-yl-methanone | CHEMBL24...)
Affinity DataIC50: 134nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO cells after 4 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207772(adamantan-1-yl-piperidin-1-yl-methanone | CHEMBL24...)
Affinity DataIC50: 193nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207799(adamantan-2-yl-piperidin-1-yl-methanone | CHEMBL24...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mouse)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207787(adamantan-1-yl-(octahydro-isoquinolin-2-yl)-methan...)
Affinity DataIC50: 230nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO cells after 4 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mouse)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207776(adamantan-1-yl-(4-ethyl-piperazin-1-yl)-methanone ...)
Affinity DataIC50: 300nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO cells after 4 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mouse)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207795(adamantan-1-yl-(3,4-dihydro-2H-quinolin-1-yl)-meth...)
Affinity DataIC50: 481nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO cells after 4 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mouse)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207767(adamantan-1-yl-[4-(2-hydroxy-ethyl)-piperazin-1-yl...)
Affinity DataIC50: 494nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO cells after 4 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207788((3R,5R)-adamantan-1-yl(pyrrolidin-1-yl)methanone |...)
Affinity DataIC50: 498nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207760([4-(2-hydroxy-ethyl)-piperazin-1-yl]-(3-p-tolyl-ad...)
Affinity DataIC50: 498nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207770((4-ethyl-piperazin-1-yl)-[3-(4-methoxy-phenyl)-ada...)
Affinity DataIC50: 600nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207800(adamantan-1-yl-(4-methyl-piperazin-1-yl)-methanone...)
Affinity DataIC50: 700nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207776(adamantan-1-yl-(4-ethyl-piperazin-1-yl)-methanone ...)
Affinity DataIC50: 756nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207787(adamantan-1-yl-(octahydro-isoquinolin-2-yl)-methan...)
Affinity DataIC50: 846nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207790((3-benzyl-adamantan-1-yl)-(4-ethyl-piperazin-1-yl)...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mouse)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207757((4-tert-butylcyclohexyl)(4-ethylpiperazin-1-yl)met...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO cells after 4 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207767(adamantan-1-yl-[4-(2-hydroxy-ethyl)-piperazin-1-yl...)
Affinity DataIC50: 1.47E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207789((4-benzyl-piperazin-1-yl)-(3-p-tolyl-adamantan-1-y...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207795(adamantan-1-yl-(3,4-dihydro-2H-quinolin-1-yl)-meth...)
Affinity DataIC50: 1.86E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207769((4-phenethyl-piperazin-1-yl)-(3-p-tolyl-adamantan-...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207781(phenyl-[4-(3-p-tolyl-adamantane-1-carbonyl)-pipera...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207773([4-(2-methoxy-ethyl)-piperazin-1-yl]-(3-p-tolyl-ad...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207765(2-adamantan-1-yl-1-(4-ethyl-piperazin-1-yl)-ethano...)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207786(adamantan-1-yl-(3,4-dihydro-1H-isoquinolin-2-yl)-m...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207797(1-(4-ethylpiperazin-1-yl)-2-phenylethanone | CHEMB...)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207774(adamantan-1-yl-(4-pyridin-4-ylmethyl-piperazin-1-y...)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207803(adamantan-1-yl-(4-benzyl-piperazin-1-yl)-methanone...)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207784((3-hydroxy-adamantan-1-yl)-piperidin-1-yl-methanon...)
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207777((4-phenyl-piperazin-1-yl)-(3-p-tolyl-adamantan-1-y...)
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207756((4-phenylmethanesulfonyl-piperazin-1-yl)-(3-p-toly...)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207779((4-pyridin-4-ylmethyl-piperazin-1-yl)-(3-p-tolyl-a...)
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207783(adamantan-1-yl-piperazin-1-yl-methanone | CHEMBL39...)
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207766(3-methyl-2-[4-(3-p-tolyl-adamantane-1-carbonyl)-pi...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207780((4-ethylpiperazin-1-yl)(1-(4-fluorophenyl)cyclopen...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207792(adamantan-1-yl-[4-(2-methoxy-ethyl)-piperazin-1-yl...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207763(adamantan-1-yl-(4-phenylmethanesulfonyl-piperazin-...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207801((4-ethylpiperazin-1-yl)(3-methyl-1H-inden-2-yl)met...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207757((4-tert-butylcyclohexyl)(4-ethylpiperazin-1-yl)met...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207758(2-[4-(adamantane-1-carbonyl)-piperazin-1-yl]-3-met...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207798([4-(adamantane-1-carbonyl)-piperazin-1-yl]-phenyl-...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207761(phenyl-[4-(3-p-tolyl-adamantane-1-carbonyl)-pipera...)
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207785(bicyclo[2.2.1]heptan-2-yl(4-ethylpiperazin-1-yl)me...)
Affinity DataIC50: 4.40E+4nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207771(adamantan-1-yl-(4-phenethyl-piperazin-1-yl)-methan...)
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207794(3-cyclohexyl-1-(4-ethylpiperazin-1-yl)propan-1-one...)
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207775((4-ethyl-piperazin-1-yl)-(3-hydroxy-adamantan-1-yl...)
Affinity DataIC50: 5.30E+4nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207802(cyclohexyl(4-ethylpiperazin-1-yl)methanone | CHEMB...)
Affinity DataIC50: 5.30E+4nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207778((4-benzenesulfonyl-piperazin-1-yl)-(3-p-tolyl-adam...)
Affinity DataIC50: 6.40E+4nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
University of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207796(1-(4-ethylpiperazin-1-yl)-2,2-dimethylpropan-1-one...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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