Compile Data Set for Download or QSAR
maximum 50k data
Found 42 Enz. Inhib. hit(s) with all data for entry = 50019857
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208409((S)-1-((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208409((S)-1-((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino...)
Affinity DataIC50:  26nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208401(5-((1,4-diazepan-1-yl)methyl)-N-(1-(3-fluorobenzyl...)
Affinity DataIC50:  27nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208401(5-((1,4-diazepan-1-yl)methyl)-N-(1-(3-fluorobenzyl...)
Affinity DataIC50:  33nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208410(1-((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino)pyr...)
Affinity DataIC50:  39nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208412(2-((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino)pyr...)
Affinity DataIC50:  45nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208412(2-((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino)pyr...)
Affinity DataIC50:  47nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208402(1-((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino)pyr...)
Affinity DataIC50:  63nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208402(1-((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino)pyr...)
Affinity DataIC50:  68nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208397(CHEMBL398793 | N-(1-(3-fluorobenzyl)-1H-indazol-5-...)
Affinity DataIC50:  74nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208416((R)-1-((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino...)
Affinity DataIC50:  76nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208399(CHEMBL231875 | N-(1-(3-fluorobenzyl)-1H-indazol-5-...)
Affinity DataIC50:  81nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50204124(CHEMBL427671 | N-(1-(3-fluorobenzyl)-1H-indazol-5-...)
Affinity DataIC50:  81nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50204124(CHEMBL427671 | N-(1-(3-fluorobenzyl)-1H-indazol-5-...)
Affinity DataIC50:  88nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208399(CHEMBL231875 | N-(1-(3-fluorobenzyl)-1H-indazol-5-...)
Affinity DataIC50:  90nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208403(1-((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino)pyr...)
Affinity DataIC50:  110nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208413(2-(((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino)py...)
Affinity DataIC50:  110nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208413(2-(((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino)py...)
Affinity DataIC50:  110nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208407(CHEMBL232082 | N-(1-(3-fluorobenzyl)-1H-indazol-5-...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208408(CHEMBL400413 | N-(1-(3-fluorobenzyl)-1H-indazol-5-...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208398(CHEMBL234577 | N-(1-(3-fluorobenzyl)-1H-indazol-5-...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208397(CHEMBL398793 | N-(1-(3-fluorobenzyl)-1H-indazol-5-...)
Affinity DataIC50:  130nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208398(CHEMBL234577 | N-(1-(3-fluorobenzyl)-1H-indazol-5-...)
Affinity DataIC50:  130nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208406(1-((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino)pyr...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208414(CHEMBL392774 | N-(1-(3-fluorobenzyl)-1H-indazol-5-...)
Affinity DataIC50:  170nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208407(CHEMBL232082 | N-(1-(3-fluorobenzyl)-1H-indazol-5-...)
Affinity DataIC50:  170nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208414(CHEMBL392774 | N-(1-(3-fluorobenzyl)-1H-indazol-5-...)
Affinity DataIC50:  190nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208416((R)-1-((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208415(4-((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino)pyr...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208408(CHEMBL400413 | N-(1-(3-fluorobenzyl)-1H-indazol-5-...)
Affinity DataIC50:  210nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208403(1-((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino)pyr...)
Affinity DataIC50:  220nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208411(1-((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino)pyr...)
Affinity DataIC50:  240nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208406(1-((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino)pyr...)
Affinity DataIC50:  310nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208415(4-((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino)pyr...)
Affinity DataIC50:  350nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208405(CHEMBL391675 | N-(1-(3-fluorobenzyl)-1H-indazol-5-...)
Affinity DataIC50:  360nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208405(CHEMBL391675 | N-(1-(3-fluorobenzyl)-1H-indazol-5-...)
Affinity DataIC50:  500nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208400(1-(4-((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino)...)
Affinity DataIC50:  610nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208400(1-(4-((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino)...)
Affinity DataIC50:  710nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208411(1-((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino)pyr...)
Affinity DataIC50:  750nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208410(1-((4-(1-(3-fluorobenzyl)-1H-indazol-5-ylamino)pyr...)
Affinity DataIC50:  780nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208404(CHEMBL231663 | methyl 1-((4-(1-(3-fluorobenzyl)-1H...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50208404(CHEMBL231663 | methyl 1-((4-(1-(3-fluorobenzyl)-1H...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of human HER2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed