Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50038474
TargetTyrosine-protein kinase ABL1(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50376901(TG-100855 | CHEMBL256101)
Affinity DataKi:  2.04nMAssay Description:Inhibition of Abl by luminescence based kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50376901(TG-100855 | CHEMBL256101)
Affinity DataKi:  4.19nMAssay Description:Inhibition of Lyn by luminescence based kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Yes(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50376901(TG-100855 | CHEMBL256101)
Affinity DataKi:  5.97nMAssay Description:Inhibition of Yes by luminescence based kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50376901(TG-100855 | CHEMBL256101)
Affinity DataKi:  7.22nMAssay Description:Inhibition of Src by luminescence based kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetEphrin type-B receptor 4(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50376901(TG-100855 | CHEMBL256101)
Affinity DataKi:  7.27nMAssay Description:Inhibition of EphB4 by luminescence based kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50376901(TG-100855 | CHEMBL256101)
Affinity DataKi:  11.7nMAssay Description:Inhibition of Lck by luminescence based kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Yes(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50198782(US8481536, 367 | 7-(2,6-dichlorophenyl)-5-methyl-N...)
Affinity DataKi:  12.9nMAssay Description:Inhibition of Yes by luminescence based kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50198782(US8481536, 367 | 7-(2,6-dichlorophenyl)-5-methyl-N...)
Affinity DataKi:  19.4nMAssay Description:Inhibition of Abl by luminescence based kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50198782(US8481536, 367 | 7-(2,6-dichlorophenyl)-5-methyl-N...)
Affinity DataKi:  25.9nMAssay Description:Inhibition of Lyn by luminescence based kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50198782(US8481536, 367 | 7-(2,6-dichlorophenyl)-5-methyl-N...)
Affinity DataKi:  28.1nMAssay Description:Inhibition of Src by luminescence based kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50198782(US8481536, 367 | 7-(2,6-dichlorophenyl)-5-methyl-N...)
Affinity DataKi:  29.4nMAssay Description:Inhibition of Lck by luminescence based kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetEphrin type-B receptor 4(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50198782(US8481536, 367 | 7-(2,6-dichlorophenyl)-5-methyl-N...)
Affinity DataKi:  63.8nMAssay Description:Inhibition of EphB4 by luminescence based kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed