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Found 12 Enz. Inhib. hit(s) with all data for entry = 50003824
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50209771(3,4-dihydroquinolin-2(1H)-one | CHEMBL388582 | Dih...)
Affinity DataIC50:  0.740nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 2 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50045333(CHEBI:90705 | SB-203580)
Affinity DataIC50:  56nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50476266(CHEMBL388106)
Affinity DataIC50:  500nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50476263(CHEMBL388130)
Affinity DataIC50:  900nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50476272(CHEMBL227884)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50476269(CHEMBL226972)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50476264(CHEMBL425494)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50476271(CHEMBL228075)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50476270(CHEMBL389508)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50476267(CHEMBL227692)
Affinity DataIC50:  1.75E+4nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50476268(CHEMBL227609)
Affinity DataIC50:  1.81E+4nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50476265(CHEMBL375948)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed