Compile Data Set for Download or QSAR
maximum 50k data
Found 227 Enz. Inhib. hit(s) with all data for entry = 50020213
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211341(5-bromo-6-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphen...)
Affinity DataKi:  0.140nMAssay Description:Binding affinity to human cloned adrenergic alpha1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50060964((R)-5-(2-((2-(2-ethoxyphenoxy)ethyl)amino)propyl)-...)
Affinity DataKi:  0.190nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50060964((R)-5-(2-((2-(2-ethoxyphenoxy)ethyl)amino)propyl)-...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to human cloned adrenergic alpha1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211318(3-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphe...)
Affinity DataKi:  0.560nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211342(2,4-dichloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)p...)
Affinity DataKi:  0.640nMAssay Description:Binding affinity to human cloned adrenergic alpha1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211328(3-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piper...)
Affinity DataKi:  0.730nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211320(2-cyano-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)pipera...)
Affinity DataKi:  0.770nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211356(5-bromo-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)pipera...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity to human cloned adrenergic alpha1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211350(2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piper...)
Affinity DataKi:  0.880nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211319(CHEMBL233623 | N-((1r,4r)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211336(CHEMBL234422 | N-((1r,4r)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211345(CHEMBL232593 | N-((1r,4r)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211329(CHEMBL234649 | N-((1s,4s)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211346(4-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piper...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211357(CHEMBL233592 | N-((1s,4s)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to human cloned adrenergic alpha1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211323(3-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piper...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211327(4-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphe...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to human cloned adrenergic alpha1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211356(5-bromo-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)pipera...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211348(2,4-dichloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)p...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211358(CHEMBL234232 | N-((1r,4r)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity to human dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50060964((R)-5-(2-((2-(2-ethoxyphenoxy)ethyl)amino)propyl)-...)
Affinity DataKi:  2nMAssay Description:Binding affinity to human cloned adrenergic alpha1B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211312(CHEMBL236830 | N-((1s,4s)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity to human cloned adrenergic alpha1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211307(CHEMBL429623 | N-((1s,4s)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity to human cloned adrenergic alpha1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211320(2-cyano-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)pipera...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity to human dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211316(2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piper...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity to human cloned adrenergic alpha1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211349(CHEMBL232592 | N-((1s,4s)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity to human cloned adrenergic alpha1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211351(CHEMBL234669 | N-((1r,4r)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  2.70nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211335(4-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphe...)
Affinity DataKi:  3nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211320(2-cyano-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)pipera...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity to human cloned adrenergic alpha1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211343(3-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piper...)
Affinity DataKi:  3.30nMAssay Description:Binding affinity to human cloned adrenergic alpha1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211353(CHEMBL236617 | N-((1s,4s)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  3.40nMAssay Description:Binding affinity to human cloned adrenergic alpha1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211347(5-bromo-6-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphen...)
Affinity DataKi:  3.5nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211343(3-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piper...)
Affinity DataKi:  3.5nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211329(CHEMBL234649 | N-((1s,4s)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  3.60nMAssay Description:Binding affinity to human cloned adrenergic alpha1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211340(5-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piper...)
Affinity DataKi:  3.80nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211337(CHEMBL234650 | N-((1r,4r)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  3.90nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211307(CHEMBL429623 | N-((1s,4s)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  4.30nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211342(2,4-dichloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)p...)
Affinity DataKi:  4.5nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211325(4-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piper...)
Affinity DataKi:  4.80nMAssay Description:Binding affinity to human cloned adrenergic alpha1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211353(CHEMBL236617 | N-((1s,4s)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  4.80nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211359(CHEMBL232607 | N-((1s,4s)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  4.90nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211315(CHEMBL234854 | N-((1s,4s)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  5nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211333(5-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piper...)
Affinity DataKi:  5nMAssay Description:Binding affinity to human cloned adrenergic alpha1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211334(CHEMBL236832 | N-((1s,4s)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  5.10nMAssay Description:Binding affinity to human cloned adrenergic alpha1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211317(CHEMBL391107 | N-((1s,4s)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  5.20nMAssay Description:Binding affinity to human cloned adrenergic alpha1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211321(CHEMBL391016 | N-((1r,4r)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  5.5nMAssay Description:Binding affinity to human cloned adrenergic alpha1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211325(4-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piper...)
Affinity DataKi:  5.60nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211316(2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piper...)
Affinity DataKi:  5.60nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211321(CHEMBL391016 | N-((1r,4r)-4-(4-(2-isopropoxyphenyl...)
Affinity DataKi:  5.80nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50211333(5-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piper...)
Affinity DataKi:  6nMAssay Description:Binding affinity to human cloned adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 227 total ) | Next | Last >>
Jump to: