Compile Data Set for Download or QSAR
maximum 50k data
Found 63 Enz. Inhib. hit(s) with all data for entry = 50037894
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50370986(CHEMBL1203946)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]8-OH-DPAT from rat brain 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213571(7-{4-[4-(3-chlorophenyl)-piperazin-1-yl]-butyl}-8-...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]8-OH-DPAT from rat brain 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213587(7-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-8...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]8-OH-DPAT from rat brain 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213571(7-{4-[4-(3-chlorophenyl)-piperazin-1-yl]-butyl}-8-...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]ketanserin from rat brain 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213576(7-{4-[4-(2-methoxyphenyl)-piperazin-1-yl]-butyl}-8...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]8-OH-DPAT from rat brain 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213577(7-{3-[4-(3-chlorophenyl)-piperazin-1-yl]-propyl}-8...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]ketanserin from rat brain 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213578(7-{3-[4-(3-chlorophenyl)-piperazin-1-yl]-propyl}-8...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]ketanserin from rat brain 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213587(7-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-8...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]ketanserin from rat brain 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213571(7-{4-[4-(3-chlorophenyl)-piperazin-1-yl]-butyl}-8-...)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor in Wistar rat hypothalamic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213585(7-[3-(4-phenylpiperazin-1-yl)-propyl]-8-propoxy-1,...)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]ketanserin from rat brain 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50370986(CHEMBL1203946)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor in Wistar rat hypothalamic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213588(7-[4-(4-phenylpiperazin-1-yl)-butyl]-8-propoxy-1,3...)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]ketanserin from rat brain 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213581(7-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)-butyl]-8...)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor in Wistar rat hypothalamic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213580(7-{3-[4-(3-chlorophenyl)-piperazin-1-yl]-propyl}-1...)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]ketanserin from rat brain 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213572(7-{4-[4-(3-chlorophenyl)-piperazin-1-yl]-butyl}-1,...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]ketanserin from rat brain 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213584(7-[4-(4-phenylpiperazin-1-yl)-butyl]-8-ethoxy-1,3-...)
Affinity DataKi:  67nMAssay Description:Displacement of [3H]8-OH-DPAT from rat brain 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213579(7-{3-[4-(2-methoxyphenyl)-piperazin-1-yl]-propyl}-...)
Affinity DataKi:  83nMAssay Description:Displacement of [3H]8-OH-DPAT from rat brain 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213570(7-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)-butyl]-8...)
Affinity DataKi:  83nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor in Wistar rat hypothalamic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213587(7-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-8...)
Affinity DataKi:  125nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor in Wistar rat hypothalamic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213588(7-[4-(4-phenylpiperazin-1-yl)-butyl]-8-propoxy-1,3...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]8-OH-DPAT from rat brain 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213577(7-{3-[4-(3-chlorophenyl)-piperazin-1-yl]-propyl}-8...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor in Wistar rat hypothalamic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213584(7-[4-(4-phenylpiperazin-1-yl)-butyl]-8-ethoxy-1,3-...)
Affinity DataKi:  131nMAssay Description:Displacement of [3H]ketanserin from rat brain 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213576(7-{4-[4-(2-methoxyphenyl)-piperazin-1-yl]-butyl}-8...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]ketanserin from rat brain 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213576(7-{4-[4-(2-methoxyphenyl)-piperazin-1-yl]-butyl}-8...)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor in Wistar rat hypothalamic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213575(7-[3-(4-phenylpiperazin-1-yl)-propyl]-8-ethoxy-1,3...)
Affinity DataKi:  176nMAssay Description:Displacement of [3H]ketanserin from rat brain 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213577(7-{3-[4-(3-chlorophenyl)-piperazin-1-yl]-propyl}-8...)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]8-OH-DPAT from rat brain 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213584(7-[4-(4-phenylpiperazin-1-yl)-butyl]-8-ethoxy-1,3-...)
Affinity DataKi:  197nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor in Wistar rat hypothalamic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213582(7-[3-(4-phenylpiperazin-1-yl)-propyl]-1,3-dimethyl...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]ketanserin from rat brain 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50370986(CHEMBL1203946)
Affinity DataKi:  253nMAssay Description:Displacement of [3H]ketanserin from rat brain 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213572(7-{4-[4-(3-chlorophenyl)-piperazin-1-yl]-butyl}-1,...)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]8-OH-DPAT from rat brain 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213578(7-{3-[4-(3-chlorophenyl)-piperazin-1-yl]-propyl}-8...)
Affinity DataKi:  267nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor in Wistar rat hypothalamic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213578(7-{3-[4-(3-chlorophenyl)-piperazin-1-yl]-propyl}-8...)
Affinity DataKi:  288nMAssay Description:Displacement of [3H]8-OH-DPAT from rat brain 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213590(7-{3-[4-(2-methoxyphenyl)-piperazin-1-yl]-propyl}-...)
Affinity DataKi:  314nMAssay Description:Displacement of [3H]8-OH-DPAT from rat brain 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213590(7-{3-[4-(2-methoxyphenyl)-piperazin-1-yl]-propyl}-...)
Affinity DataKi:  328nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor in Wistar rat hypothalamic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213581(7-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)-butyl]-8...)
Affinity DataKi:  332nMAssay Description:Displacement of [3H]8-OH-DPAT from rat brain 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213579(7-{3-[4-(2-methoxyphenyl)-piperazin-1-yl]-propyl}-...)
Affinity DataKi:  410nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor in Wistar rat hypothalamic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213570(7-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)-butyl]-8...)
Affinity DataKi:  430nMAssay Description:Displacement of [3H]8-OH-DPAT from rat brain 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213575(7-[3-(4-phenylpiperazin-1-yl)-propyl]-8-ethoxy-1,3...)
Affinity DataKi:  477nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor in Wistar rat hypothalamic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213590(7-{3-[4-(2-methoxyphenyl)-piperazin-1-yl]-propyl}-...)
Affinity DataKi:  540nMAssay Description:Displacement of [3H]ketanserin from rat brain 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213586(7-[4-(4-phenylpiperazin-1-yl)-butyl]-1,3-dimethyl-...)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]ketanserin from rat brain 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213589(7-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-8...)
Affinity DataKi:  590nMAssay Description:Displacement of [3H]ketanserin from rat brain 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213588(7-[4-(4-phenylpiperazin-1-yl)-butyl]-8-propoxy-1,3...)
Affinity DataKi:  680nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor in Wistar rat hypothalamic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213585(7-[3-(4-phenylpiperazin-1-yl)-propyl]-8-propoxy-1,...)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]8-OH-DPAT from rat brain 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213581(7-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)-butyl]-8...)
Affinity DataKi:  920nMAssay Description:Displacement of [3H]ketanserin from rat brain 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213579(7-{3-[4-(2-methoxyphenyl)-piperazin-1-yl]-propyl}-...)
Affinity DataKi:  980nMAssay Description:Displacement of [3H]ketanserin from rat brain 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213585(7-[3-(4-phenylpiperazin-1-yl)-propyl]-8-propoxy-1,...)
Affinity DataKi:  980nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor in Wistar rat hypothalamic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213573(7-[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)-propyl]-...)
Affinity DataKi:  1.01E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from rat brain 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213589(7-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-8...)
Affinity DataKi:  1.07E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from rat brain 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213580(7-{3-[4-(3-chlorophenyl)-piperazin-1-yl]-propyl}-1...)
Affinity DataKi:  1.11E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from rat brain 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50213575(7-[3-(4-phenylpiperazin-1-yl)-propyl]-8-ethoxy-1,3...)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from rat brain 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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