Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50020583
TargetCholecystokinin receptor type A(Human)
Istituto Di Biostrutture E Bioimmagini-Cnr

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50215386BDBM50215386((S)-5-(2-((S)-1-((S)-1-((S)-1-((S)-1-(3-amino-1-((...)
Affinity DataIC50: 32nMAssay Description:Displacement of [111In]DTPA-Glu-Gly-[Tyr27(SO3H)]-CCK8 from human CCK1 receptor expressed in A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
Istituto Di Biostrutture E Bioimmagini-Cnr

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50215383BDBM50215383((3S)-3-amino-3-{[(1S)-1-{[(1S)-1-{[(5S,8S,11S)-11-...)
Affinity DataIC50: 6.45E+3nMAssay Description:Displacement of [111In]DTPA-Glu-Gly-[Tyr27(SO3H)]-CCK8 from human CCK1 receptor expressed in A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
Istituto Di Biostrutture E Bioimmagini-Cnr

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50215381BDBM50215381((3S)-3-amino-3-{[(1S)-1-{[(1S)-1-{[(2S,5S,8S)-11-[...)
Affinity DataIC50: 6.94E+3nMAssay Description:Displacement of [111In]DTPA-Glu-Gly-[Tyr27(SO3H)]-CCK8 from human CCK1 receptor expressed in A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
Istituto Di Biostrutture E Bioimmagini-Cnr

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50215385BDBM50215385((3S)-3-amino-3-{[(1S)-1-{[(1S)-1-{[(2S,5S,8S,11S)-...)
Affinity DataIC50: 7.20E+3nMAssay Description:Displacement of [111In]DTPA-Glu-Gly-[Tyr27(SO3H)]-CCK8 from human CCK1 receptor expressed in A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
Istituto Di Biostrutture E Bioimmagini-Cnr

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50215388BDBM50215388((3S)-3-amino-3-{[(1S)-1-{[(1S)-1-{[(2S,5S,8S)-11-[...)
Affinity DataIC50: 7.46E+3nMAssay Description:Displacement of [111In]DTPA-Glu-Gly-[Tyr27(SO3H)]-CCK8 from human CCK1 receptor expressed in A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
Istituto Di Biostrutture E Bioimmagini-Cnr

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50215379BDBM50215379((3S)-3-amino-3-{[(1S)-1-{[(1S)-1-{[(3S,6S,9S,12S,1...)
Affinity DataIC50: 1.50E+4nMAssay Description:Displacement of [111In]DTPA-Glu-Gly-[Tyr27(SO3H)]-CCK8 from human CCK1 receptor expressed in A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
Istituto Di Biostrutture E Bioimmagini-Cnr

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50215384BDBM50215384((3S)-3-amino-3-{[(1S)-1-{[(1S)-1-{[(2S,5S,8S,11S)-...)
Affinity DataIC50: 2.48E+4nMAssay Description:Displacement of [111In]DTPA-Glu-Gly-[Tyr27(SO3H)]-CCK8 from human CCK1 receptor expressed in A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
Istituto Di Biostrutture E Bioimmagini-Cnr

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50215387BDBM50215387((3S)-3-amino-3-{[(1S)-1-{[(1S)-1-{[(2S,5S,8S,11S)-...)
Affinity DataIC50: 2.63E+4nMAssay Description:Displacement of [111In]DTPA-Glu-Gly-[Tyr27(SO3H)]-CCK8 from human CCK1 receptor expressed in A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
Istituto Di Biostrutture E Bioimmagini-Cnr

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50215380BDBM50215380((3S)-3-amino-3-{[(1S)-1-{[(1S)-1-{[(3S,6S,9S,12S)-...)
Affinity DataIC50: 2.67E+4nMAssay Description:Displacement of [111In]DTPA-Glu-Gly-[Tyr27(SO3H)]-CCK8 from human CCK1 receptor expressed in A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
Istituto Di Biostrutture E Bioimmagini-Cnr

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50215382BDBM50215382((3S)-3-amino-3-{[(1S)-1-{[(1S)-1-{[(3S,6S,9S,12S,1...)
Affinity DataIC50: 1.00E+6nMAssay Description:Displacement of [111In]DTPA-Glu-Gly-[Tyr27(SO3H)]-CCK8 from human CCK1 receptor expressed in A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed