Compile Data Set for Download or QSAR
maximum 50k data
Found 63 Enz. Inhib. hit(s) with all data for entry = 50020921
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50152456((S)-3-{3-[4-(3-Acetylamino-phenyl)-piperidin-1-yl]...)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219047(CHEMBL245231 | N-(3-(1-(4-(3,4-difluorophenoxy)ben...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219053(CHEMBL242004 | N-(3-{1-4-(3,4-difluorophenoxy)benz...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219062(CHEMBL394569 | N-(3-{1-[4-(4-chlorophenyl)-4-oxobu...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219064(CHEMBL245010 | N-(3-{1-[4-(4-chlorophenoxy)benzyl]...)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219050(CHEMBL389129 | N-(3-{1-[4-(3,4-dichlorophenoxy)ben...)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219054(2-methyl-N-{3-[1-(4-phenoxybenzyl)-4-piperidinyl]p...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219055(CHEMBL244791 | N-(3-{1-[3-(3,4-dichlorophenoxy)ben...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219066(CHEMBL244578 | N-(3-{1-[3-(4-chlorophenoxy)benzyl]...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219045(CHEMBL242003 | N-(5-{1-[4-(3,4-difluorophenoxy)ben...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219063(2-methyl-N-{3-[1-(3-phenoxybenzyl)-4-piperidinyl]p...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219065(2-methyl-N-(3-{1-[3-(4-methylphenoxy)benzyl]-4-pip...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219051(CHEMBL245229 | N-(3-{1-[4-(4-methoxyphenoxy)benzyl...)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50152456((S)-3-{3-[4-(3-Acetylamino-phenyl)-piperidin-1-yl]...)
Affinity DataKi:  40nMAssay Description:Displacement of [125I]HEAT from human recombinant adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219059(CHEMBL390212 | N-(3-{1-[3-(4-methoxyphenoxy)benzyl...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219052(2-methyl-N-[3-(1-{3-[3-(trifluoromethyl)phenoxy]be...)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219061(CHEMBL243794 | N-(3-{1-[4-(4-chlorophenyl)-4-oxobu...)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219048(CHEMBL244372 | N-(3-{1-[4-(4-chlorophenyl)-4-oxobu...)
Affinity DataKi:  84nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219058(CHEMBL244004 | N-(3-{1-[4-(3,4-dimethylphenyl)-4-o...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219064(CHEMBL245010 | N-(3-{1-[4-(4-chlorophenoxy)benzyl]...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219054(2-methyl-N-{3-[1-(4-phenoxybenzyl)-4-piperidinyl]p...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219068(CHEMBL245008 | N-(3-{1-[3-(3,5-dichlorophenoxy)ben...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219049(1-(4-Chloro-phenyl)-4-[4-(4-chloro-phenyl)-4-hydro...)
Affinity DataKi:  150nMAssay Description:Displacement of [125I]HEAT from human recombinant adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219053(CHEMBL242004 | N-(3-{1-4-(3,4-difluorophenoxy)benz...)
Affinity DataKi:  180nMAssay Description:Displacement of [125I]HEAT from human recombinant adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219049(1-(4-Chloro-phenyl)-4-[4-(4-chloro-phenyl)-4-hydro...)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219056(CHEMBL244163 | N-(3-{1-[4-(4-chlorophenyl)-4-oxobu...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219047(CHEMBL245231 | N-(3-(1-(4-(3,4-difluorophenoxy)ben...)
Affinity DataKi:  200nMAssay Description:Displacement of [125I]HEAT from human recombinant adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219049(1-(4-Chloro-phenyl)-4-[4-(4-chloro-phenyl)-4-hydro...)
Affinity DataKi:  350nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219046(CHEMBL395788 | N-{3-[1-(4-oxo-4-phenylbutyl)-4-pip...)
Affinity DataKi:  350nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219057(CHEMBL395789 | N-(3-{1-[4-(4-methylphenyl)-4-oxobu...)
Affinity DataKi:  360nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219045(CHEMBL242003 | N-(5-{1-[4-(3,4-difluorophenoxy)ben...)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219047(CHEMBL245231 | N-(3-(1-(4-(3,4-difluorophenoxy)ben...)
Affinity DataKi:  470nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219060(CHEMBL244003 | N-(3-{1-[4-oxo-4-(4-phenoxyphenyl)b...)
Affinity DataKi:  490nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219067(CHEMBL244576 | N-(3-{1-[3-(4-tert-butylphenoxy)ben...)
Affinity DataKi:  540nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219062(CHEMBL394569 | N-(3-{1-[4-(4-chlorophenyl)-4-oxobu...)
Affinity DataKi:  610nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219048(CHEMBL244372 | N-(3-{1-[4-(4-chlorophenyl)-4-oxobu...)
Affinity DataKi:  780nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219059(CHEMBL390212 | N-(3-{1-[3-(4-methoxyphenoxy)benzyl...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219045(CHEMBL242003 | N-(5-{1-[4-(3,4-difluorophenoxy)ben...)
Affinity DataKi:  1.01E+3nMAssay Description:Displacement of [125I]HEAT from human recombinant adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219065(2-methyl-N-(3-{1-[3-(4-methylphenoxy)benzyl]-4-pip...)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219061(CHEMBL243794 | N-(3-{1-[4-(4-chlorophenyl)-4-oxobu...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219051(CHEMBL245229 | N-(3-{1-[4-(4-methoxyphenoxy)benzyl...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50152456((S)-3-{3-[4-(3-Acetylamino-phenyl)-piperidin-1-yl]...)
Affinity DataKi:  2.80E+3nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219050(CHEMBL389129 | N-(3-{1-[4-(3,4-dichlorophenoxy)ben...)
Affinity DataKi:  2.90E+3nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219058(CHEMBL244004 | N-(3-{1-[4-(3,4-dimethylphenyl)-4-o...)
Affinity DataKi:  6.10E+3nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219053(CHEMBL242004 | N-(3-{1-4-(3,4-difluorophenoxy)benz...)
Affinity DataKi:  7.40E+3nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219050(CHEMBL389129 | N-(3-{1-[4-(3,4-dichlorophenoxy)ben...)
Affinity DataKi:  3.40E+4nMAssay Description:Displacement of [125I]HEAT from human recombinant adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219062(CHEMBL394569 | N-(3-{1-[4-(4-chlorophenyl)-4-oxobu...)
Affinity DataIC50:  72nMAssay Description:Antagonist activity at rat MCH1 receptor expressed in HEK293 cells by FLIPR calcium mobility assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219047(CHEMBL245231 | N-(3-(1-(4-(3,4-difluorophenoxy)ben...)
Affinity DataIC50:  110nMAssay Description:Antagonist activity at rat MCH1 receptor expressed in HEK293 cells by FLIPR calcium mobility assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219053(CHEMBL242004 | N-(3-{1-4-(3,4-difluorophenoxy)benz...)
Affinity DataIC50:  230nMAssay Description:Antagonist activity at rat MCH1 receptor expressed in HEK293 cells by FLIPR calcium mobility assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50219054(2-methyl-N-{3-[1-(4-phenoxybenzyl)-4-piperidinyl]p...)
Affinity DataIC50:  320nMAssay Description:Antagonist activity at rat MCH1 receptor expressed in HEK293 cells by FLIPR calcium mobility assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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