Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50037962
TargetMetabotropic glutamate receptor 1(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM17657(L-Glutamic acid | L-Glu | (2S)-2-aminopentanedioic...)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM17657(L-Glutamic acid | L-Glu | (2S)-2-aminopentanedioic...)
Affinity DataKi:  390nMAssay Description:Binding affinity to mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM17657(L-Glutamic acid | L-Glu | (2S)-2-aminopentanedioic...)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM17657(L-Glutamic acid | L-Glu | (2S)-2-aminopentanedioic...)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220148((2S,1'R,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi:  3.40E+4nMAssay Description:Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220148((2S,1'R,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi:  4.90E+4nMAssay Description:Binding affinity to mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220147(L-homocysteic acid | L-Homocysteate | (S)-2-amino-...)
Affinity DataKi:  5.30E+4nMAssay Description:Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220147(L-homocysteic acid | L-Homocysteate | (S)-2-amino-...)
Affinity DataKi:  5.40E+4nMAssay Description:Binding affinity to mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220154((2R,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi:  5.50E+4nMAssay Description:Binding affinity to mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220150((2R,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi:  6.70E+4nMAssay Description:Binding affinity to mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220149((2S,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi:  7.70E+4nMAssay Description:Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220149((2S,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi:  8.10E+4nMAssay Description:Binding affinity to mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220147(L-homocysteic acid | L-Homocysteate | (S)-2-amino-...)
Affinity DataKi:  8.70E+4nMAssay Description:Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220148((2S,1'R,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi:  2.35E+5nMAssay Description:Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220150((2R,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi:  2.54E+5nMAssay Description:Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220153((2R,1'R,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220150((2R,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220145((2S,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220146((2S,1'S,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Binding affinity to mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220147(L-homocysteic acid | L-Homocysteate | (S)-2-amino-...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220150((2R,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220149((2S,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220145((2S,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Binding affinity to mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220151((2R,1'S,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Binding affinity to mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220146((2S,1'S,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220145((2S,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220146((2S,1'S,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220153((2R,1'R,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Binding affinity to mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220148((2S,1'R,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220153((2R,1'R,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220151((2R,1'S,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220151((2R,1'S,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220154((2R,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220153((2R,1'R,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220149((2S,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220151((2R,1'S,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220154((2R,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220154((2R,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220146((2S,1'S,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50220145((2S,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed