Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50021401
TargetSubstance-P receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50224198((2S,3S)-N-(2-methoxy-5-(1,1,1-trifluoro-2-methylpr...)
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at neurokinin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50224197((2S,3S)-N-(5-tert-butyl-2-methoxybenzyl)-2-phenylp...)
Affinity DataIC50: 0.600nMAssay Description:Antagonist activity at neurokinin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50160039(N-(4-tert-Butyl-phenyl)-4-(3-chloro-pyridin-2-yl)-...)
Affinity DataIC50: 37nMAssay Description:Antagonist activity at human TRPV1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50224199(4-(3-chloropyridin-2-yl)-N-(4-(1,1,1-trifluoro-2-m...)
Affinity DataIC50: 42nMAssay Description:Antagonist activity at human TRPV1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50191743(4-(3-chloropyridin-2-yl)-N-(4-(trifluoromethyl)phe...)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at human TRPV1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed