Compile Data Set for Download or QSAR
Report error Found 53 Enz. Inhib. hit(s) with all data for entry = 50025625
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7107(CHEMBL190446 | (2S)-N-(5-cyclopropyl-1H-pyrazol-3-...)
Affinity DataIC50: 2nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7111((2S)-N-(5-Cyclopropyl-1H-pyrazol-3-yl)-2-[4-(2-oxo...)
Affinity DataIC50: 2nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM50247314(N-(5-cyclopropyl-1H-pyrazol-3-yl)-2-(4-(thiophen-2...)
Affinity DataIC50: 3nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM50247290(N-(5-cyclopropyl-1H-pyrazol-3-yl)-2-(2-fluorobiphe...)
Affinity DataIC50: 4nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM50247313(N-(5-cyclopropyl-1H-pyrazol-3-yl)-2-(2-methylbiphe...)
Affinity DataIC50: 9nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7118(CHEMBL192042 | (2S)-N-(5-Cyclopropyl-1H-pyrazol-3-...)
Affinity DataIC50: 17nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7120((2S)-N-(5-Cyclopropyl-1H-pyrazol-3-yl)-2-[4-(2-oxo...)
Affinity DataIC50: 20nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7155(CHEMBL114917 | N-(5-cyclopropyl-1H-pyrazol-3-yl)-2...)
Affinity DataIC50: 29nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7128(CHEMBL115319 | 4-bromo-N-(5-cyclopropyl-1H-pyrazol...)
Affinity DataIC50: 34nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7101((2S)-N-(5-Cyclopropyl-1H-pyrazol-3-yl)-2-[4-(2-oxo...)
Affinity DataIC50: 37nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7153(N-(5-cyclopropyl-1H-pyrazol-3-yl)-2-phenylacetamid...)
Affinity DataIC50: 48nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7143(CHEMBL419753 | 4-bromo-N-(5-cyclopentyl-1H-pyrazol...)
Affinity DataIC50: 50nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7158(2-(1,1 -Biphenyl-4-yl)-N-(5-cyclopropyl-1H-pyrazol...)
Affinity DataIC50: 56nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7157(N-(5-Cyclopropyl-1H-pyrazol-3-yl)-2-(4-trifluorome...)
Affinity DataIC50: 67nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7132(CHEMBL325606 | 1-N-(5-cyclopropyl-1H-pyrazol-3-yl)...)
Affinity DataIC50: 68nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7154(CHEMBL324577 | 4-{2-[(5-Cyclopropyl-1H-pyrazol-3-y...)
Affinity DataIC50: 74nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7123((2S)-N-(5-cyclopropyl-1H-pyrazol-3-yl)-2-[4-(pyrro...)
Affinity DataIC50: 80nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7141(3,4-dichloro-N-(5-cyclopropyl-1H-pyrazol-3-yl)benz...)
Affinity DataIC50: 83nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7098((2S)-N-(5-Cyclopropyl-1H-pyrazol-3-yl)-2-phenylpro...)
Affinity DataIC50: 84nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7129(CHEMBL115264 | N-(5-Cyclopropyl-1H-pyrazol-3-yl)-4...)
Affinity DataIC50: 85nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7142(N-(5-Cyclobutyl-1H-pyrazol-3-yl)-4-bromobenzamide ...)
Affinity DataIC50: 90nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7131(4-[(5-cyclopropyl-1H-pyrazol-3-yl)carbamoyl]benzoi...)
Affinity DataIC50: 165nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7106((2R)-N-(5-cyclopropyl-1H-pyrazol-3-yl)-2-[4-(1-oxo...)
Affinity DataIC50: 170nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7148(N-(5-Isopropyl-1H-pyrazol-3-yl)-4-bromobenzamide |...)
Affinity DataIC50: 200nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7126(CS2 | N-(5-Cyclopropyl-1H-pyrazol-3-yl)butanamide ...)
Affinity DataIC50: 224nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7127(CHEMBL324942 | N-(5-cyclopropyl-1H-pyrazol-3-yl)be...)
Affinity DataIC50: 290nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7110(CHEMBL189047 | (2R)-N-(5-Cyclopropyl-1H-pyrazol-3-...)
Affinity DataIC50: 455nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7136(N-(5-Cyclopropyl-1H-pyrazol-3-yl)-3-trifluoromethy...)
Affinity DataIC50: 500nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7135(N-(5-Cyclopropyl-1H-pyrazol-3-yl)-3-methoxybenzami...)
Affinity DataIC50: 600nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7146(CHEMBL115047 | N-(5-Ethyl-1H-pyrazol-3-yl)-4-bromo...)
Affinity DataIC50: 630nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7147(N-(5-Propyl-1H-pyrazol-3-yl)-4-bromobenzamide | CH...)
Affinity DataIC50: 650nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7130(CHEMBL111897 | N-(5-Cyclopropyl-1H-pyrazol-3-yl)-4...)
Affinity DataIC50: 705nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7095((2S)-2-Amino-N-(5-cyclopropyl-1H-pyrazol-3-yl)-2-p...)
Affinity DataIC50: 960nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7133(N-(5-Cyclopropyl-1H-pyrazol-3-yl)-3-bromobenzamide...)
Affinity DataIC50: 990nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7134(3-chloro-N-(5-cyclopropyl-1H-pyrazol-3-yl)benzamid...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7137(CHEMBL116047 | 2-bromo-N-(5-cyclopropyl-1H-pyrazol...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7124(CHEMBL115125 | N-(5-Methyl-1H-pyrazol-3-yl)benzami...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7092(CHEMBL190154 | (2S)-N-(5-Cyclopropyl-1H-pyrazol-3-...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7100((2R)-N-(5-Cyclopropyl-1H-pyrazol-3-yl)-2-[4-(2-oxo...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7119(CHEMBL192179 | (2R)-N-(5-Cyclopropyl-1H-pyrazol-3-...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7097(N-(5-Cyclopropyl-1H-pyrazol-3-yl)-2-oxo-2-phenylac...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7145(4-bromo-N-(5-methyl-1H-pyrazol-3-yl)benzamide | CS...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7099(CHEMBL365988 | (2R)-N-(5-Cyclopropyl-1H-pyrazol-3-...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7117(CHEMBL365355 | (2R)-N-(5-Cyclopropyl-1H-pyrazol-3-...)
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7093(CHEMBL370036 | (2R)-N-(5-Cyclopropyl-1H-pyrazol-3-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7144(N-(5-Cycloexyl-1H-pyrazol-3-yl)-4-bromobenzamide |...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7150(4-bromo-N-(5-tert-butyl-1H-pyrazol-3-yl)benzamide ...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7152(CHEMBL420677 | N-(5-Benzyl-1H-pyrazol-3-yl)-4-brom...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7151(CHEMBL114247 | 4-bromo-N-(5-phenyl-1H-pyrazol-3-yl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Institute of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7139(CHEMBL323417 | N-(5-Cyclopropyl-1H-pyrazol-3-yl)-2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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