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Found 126 Enz. Inhib. hit(s) with all data for entry = 50038152
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372295(CHEMBL429914)
Affinity DataKi:  0.390nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372292(CHEMBL441903)
Affinity DataKi:  1.30nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372290(CHEMBL269951)
Affinity DataKi:  1.60nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372322(CHEMBL271898)
Affinity DataKi:  2.30nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372294(CHEMBL402187)
Affinity DataKi:  3.5nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372295(CHEMBL429914)
Affinity DataKi:  3.90nMAssay Description:Binding affinity at rat recombinant histamine H3 receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372291(CHEMBL271661)
Affinity DataKi:  5nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372303(CHEMBL403052)
Affinity DataKi:  5nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372304(CHEMBL257915)
Affinity DataKi:  5nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372290(CHEMBL269951)
Affinity DataKi:  5.90nMAssay Description:Binding affinity at rat recombinant histamine H3 receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372335(CHEMBL402872)
Affinity DataKi:  6nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372292(CHEMBL441903)
Affinity DataKi:  7.10nMAssay Description:Binding affinity at rat recombinant histamine H3 receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372323(CHEMBL404532)
Affinity DataKi:  8.90nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372305(CHEMBL272141)
Affinity DataKi:  10nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372329(CHEMBL270630)
Affinity DataKi:  11nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372322(CHEMBL271898)
Affinity DataKi:  12nMAssay Description:Binding affinity at rat recombinant histamine H3 receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372296(CHEMBL402377)
Affinity DataKi:  14nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372318(CHEMBL402220)
Affinity DataKi:  15nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372324(CHEMBL439429)
Affinity DataKi:  16nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372339(CHEMBL255141)
Affinity DataKi:  17nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372321(CHEMBL272988)
Affinity DataKi:  18nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372334(CHEMBL257235)
Affinity DataKi:  20nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372331(CHEMBL404834)
Affinity DataKi:  21nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372317(CHEMBL271237)
Affinity DataKi:  26nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372313(CHEMBL257911)
Affinity DataKi:  27nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372298(CHEMBL402415)
Affinity DataKi:  28nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372293(CHEMBL270410)
Affinity DataKi:  30nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372304(CHEMBL257915)
Affinity DataKi:  30nMAssay Description:Binding affinity at rat recombinant histamine H3 receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372327(CHEMBL404912)
Affinity DataKi:  31nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372315(CHEMBL257914)
Affinity DataKi:  32nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372340(CHEMBL406698)
Affinity DataKi:  33nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372310(CHEMBL408259)
Affinity DataKi:  34nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372337(CHEMBL402873)
Affinity DataKi:  34nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372329(CHEMBL270630)
Affinity DataKi:  35nMAssay Description:Binding affinity at rat recombinant histamine H3 receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372302(CHEMBL404375)
Affinity DataKi:  35nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372303(CHEMBL403052)
Affinity DataKi:  37nMAssay Description:Binding affinity at rat recombinant histamine H3 receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372291(CHEMBL271661)
Affinity DataKi:  40nMAssay Description:Binding affinity at rat recombinant histamine H3 receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372318(CHEMBL402220)
Affinity DataKi:  41nMAssay Description:Binding affinity at rat recombinant histamine H3 receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372301(CHEMBL272307)
Affinity DataKi:  41nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372336(CHEMBL271489)
Affinity DataKi:  43nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372335(CHEMBL402872)
Affinity DataKi:  43nMAssay Description:Binding affinity at rat recombinant histamine H3 receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372294(CHEMBL402187)
Affinity DataKi:  62nMAssay Description:Binding affinity at rat recombinant histamine H3 receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372323(CHEMBL404532)
Affinity DataKi:  63nMAssay Description:Binding affinity at rat recombinant histamine H3 receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372325(CHEMBL272306)
Affinity DataKi:  65nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372311(CHEMBL271722)
Affinity DataKi:  70nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372305(CHEMBL272141)
Affinity DataKi:  72nMAssay Description:Binding affinity at rat recombinant histamine H3 receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372314(CHEMBL257912)
Affinity DataKi:  81nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372339(CHEMBL255141)
Affinity DataKi:  81nMAssay Description:Binding affinity at rat recombinant histamine H3 receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372296(CHEMBL402377)
Affinity DataKi:  89nMAssay Description:Binding affinity at rat recombinant histamine H3 receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50372333(CHEMBL440996)
Affinity DataKi:  96nMAssay Description:Binding affinity at human recombinant histamine H3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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