Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50038301
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374521(CHEMBL272369)
Affinity DataIC50:  1.40nMAssay Description:Displacement of [125I]MCP1 from human CCR2 expressed in human monocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374523(CHEMBL402532)
Affinity DataIC50:  2.5nMAssay Description:Antagonist activity at human CCR2 assessed as inhibition of MCP1-induced monocyte chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374523(CHEMBL402532)
Affinity DataIC50:  4.60nMAssay Description:Displacement of [125I]MCP1 from human CCR2 expressed in human monocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374522(CHEMBL401890)
Affinity DataIC50:  115nMAssay Description:Displacement of [125I]MCP1 from human CCR2 expressed in human monocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed