Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 50038110
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371643(CHEMBL272278)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371651(CHEMBL410281)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371657(CHEMBL404370)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371653(CHEMBL255997)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50212094(3,5-dichloro-3'-fluoro-4'-((R)-1-{[1-(2,2,2-triflu...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371644(CHEMBL404484)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371658(CHEMBL270173)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371647(CHEMBL404705)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371650(CHEMBL404683)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371652(CHEMBL404280)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371656(CHEMBL401619)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371649(CHEMBL404328)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371655(CHEMBL402630)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371646(CHEMBL403202)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371659(CHEMBL269963)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371642(CHEMBL436854)
Affinity DataKi:  1.80nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371645(CHEMBL256903)
Affinity DataKi:  1.90nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371648(CHEMBL255325)
Affinity DataKi:  2.30nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371654(CHEMBL403434)
Affinity DataKi:  2.60nMAssay Description:Binding affinity to human bradykinin B1 receptor expressed in rat CNSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed