Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 50025693
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 11162BDBM11162(Triazolopiperazine Analogue 1 | (3R)-3-amino-1-[3-...)
Affinity DataIC50: 110nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245529BDBM50245529(R)-{4-[{2-[3-Amino-4-(2,4,5-trifluorophenyl)butyry...)
Affinity DataIC50: 510nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245468BDBM50245468((R)-{4-[{2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50: 690nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245275BDBM50245275((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50: 710nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245359BDBM50245359((R)-4-({2-[3-Amino-4-(2,4,5-trifluorophenyl)butyry...)
Affinity DataIC50: 770nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245404BDBM50245404((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245274BDBM50245274((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245503BDBM50245503((R)-4-[({2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245358BDBM50245358((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245321BDBM50245321((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245318BDBM50245318((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245439BDBM50245439((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245319BDBM50245319((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245469BDBM50245469((R)-{3-[{2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245438BDBM50245438((R)-{3-[({2-[3-Amino-4-(2,4,5-trifluorophenyl)buty...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245406BDBM50245406((R)-{4-[({2-[3-Amino-4-(2,4,5-trifluorophenyl)buty...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245556BDBM50245556((R)-{4-[{2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245277BDBM50245277((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245527BDBM50245527((R)-{4-[({2-[3-Amino-4-(2,4,5-trifluorophenyl)buty...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245501BDBM50245501((R)-{4-[{2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245555BDBM50245555((R)-{4-[{2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245276BDBM50245276((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245528BDBM50245528((R)-{3-[({2-[3-Amino-4-(2,4,5-trifluorophenyl)buty...)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245357BDBM50245357((R)-4-[({2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245405BDBM50245405((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245502BDBM50245502((R)-{4-[{2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245403BDBM50245403((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245553BDBM50245553((R)-{3-[{2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245470BDBM50245470((R)-{2-[{2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245320BDBM50245320((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245526BDBM50245526((R)-4-({2-[3-Amino-4-(2,4,5-trifluorophenyl)butyry...)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245360BDBM50245360((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245554BDBM50245554((R)-{2-[{2-[3-Amino-4-(2,4,5-trifluorophenyl)butyr...)
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245441BDBM50245441((R)-4-({2-[3-Amino-4-(2,4,5-trifluorophenyl)butyry...)
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245440BDBM50245440((R)-2-[3-Amino-4-(2,4,5-trifluorophenyl)butyryl]-3...)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of DPP4 in human Caco-2 cells after 60 mins by fluorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed