Compile Data Set for Download or QSAR
Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 2805
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24876(2-{5-[1-({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3...)
Affinity DataIC50: 3.80nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24883(1-[1-({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]...)
Affinity DataIC50: 4nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24875(4-{3-[1-({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3...)
Affinity DataIC50: 4.5nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24880(N-methyl-6-phenyl-7-[4-({4-[5-(pyridin-2-yl)-4H-1,...)
Affinity DataIC50: 6nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24879(6-phenyl-7-[4-({4-[5-(pyridin-2-yl)-4H-1,2,4-triaz...)
Affinity DataIC50: 6.20nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24872(5-[1-({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]...)
Affinity DataIC50: 8.5nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24873(1-({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]pyr...)
Affinity DataIC50: 9.70nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24882(7-{4-[(4-{4-amino-1H-pyrazolo[3,4-d]pyrimidin-1-yl...)
Affinity DataIC50: 14nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24867(CHEMBL252456 | 1-(2-aminophenyl)-3-[({4-[2-(methyl...)
Affinity DataIC50: 15nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24881(7-(4-{[4-(6-fluoro-1H-1,3-benzodiazol-2-yl)piperid...)
Affinity DataIC50: 18nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24877(2-(5-{1-[(4-{2-methoxy-6-phenylpyrido[2,3-d]pyrimi...)
Affinity DataIC50: 23.6nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24878(6-phenyl-7-[4-({4-[5-(pyridin-2-yl)-4H-1,2,4-triaz...)
Affinity DataIC50: 24nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24876(2-{5-[1-({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3...)
Affinity DataIC50: 26nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24868(1-({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]pyr...)
Affinity DataIC50: 29nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24879(6-phenyl-7-[4-({4-[5-(pyridin-2-yl)-4H-1,2,4-triaz...)
Affinity DataIC50: 35nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24883(1-[1-({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]...)
Affinity DataIC50: 44nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24866(5-{2-[({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d...)
Affinity DataIC50: 46nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24875(4-{3-[1-({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3...)
Affinity DataIC50: 57nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24878(6-phenyl-7-[4-({4-[5-(pyridin-2-yl)-4H-1,2,4-triaz...)
Affinity DataIC50: 59nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24865(({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]pyrim...)
Affinity DataIC50: 63nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24874(5-[1-({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]...)
Affinity DataIC50: 64nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24869(3-ethyl-1-[1-({4-[2-(methylsulfanyl)-6-phenylpyrid...)
Affinity DataIC50: 81nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24867(CHEMBL252456 | 1-(2-aminophenyl)-3-[({4-[2-(methyl...)
Affinity DataIC50: 90nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24861(({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]pyrim...)
Affinity DataIC50: 90nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24870(3-{[1-({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d...)
Affinity DataIC50: 91nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24880(N-methyl-6-phenyl-7-[4-({4-[5-(pyridin-2-yl)-4H-1,...)
Affinity DataIC50: 94.4nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24882(7-{4-[(4-{4-amino-1H-pyrazolo[3,4-d]pyrimidin-1-yl...)
Affinity DataIC50: 99nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24858([2-(1H-imidazol-4-yl)ethyl]({4-[2-(methylsulfanyl)...)
Affinity DataIC50: 99nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24877(2-(5-{1-[(4-{2-methoxy-6-phenylpyrido[2,3-d]pyrimi...)
Affinity DataIC50: 107nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24862([3-(1H-imidazol-1-yl)propyl]({4-[2-(methylsulfanyl...)
Affinity DataIC50: 137nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24859(({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]pyrim...)
Affinity DataIC50: 139nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24864([2-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]({4-[2-(m...)
Affinity DataIC50: 162nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24860(({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]pyrim...)
Affinity DataIC50: 198nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24856(3-[({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]py...)
Affinity DataIC50: 226nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24881(7-(4-{[4-(6-fluoro-1H-1,3-benzodiazol-2-yl)piperid...)
Affinity DataIC50: 239nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24872(5-[1-({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]...)
Affinity DataIC50: 267nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24871(2-acetamido-N-[1-({4-[2-(methylsulfanyl)-6-phenylp...)
Affinity DataIC50: 286nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24873(1-({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]pyr...)
Affinity DataIC50: 301nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24865(({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]pyrim...)
Affinity DataIC50: 494nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24866(5-{2-[({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d...)
Affinity DataIC50: 529nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24857([3-(4-methylpiperazin-1-yl)propyl]({4-[2-(methylsu...)
Affinity DataIC50: 765nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24868(1-({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]pyr...)
Affinity DataIC50: 928nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24861(({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]pyrim...)
Affinity DataIC50: 1.16E+3nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24858([2-(1H-imidazol-4-yl)ethyl]({4-[2-(methylsulfanyl)...)
Affinity DataIC50: 1.24E+3nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24856(3-[({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]py...)
Affinity DataIC50: 1.30E+3nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24874(5-[1-({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]...)
Affinity DataIC50: 1.30E+3nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24860(({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]pyrim...)
Affinity DataIC50: 1.38E+3nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24862([3-(1H-imidazol-1-yl)propyl]({4-[2-(methylsulfanyl...)
Affinity DataIC50: 1.51E+3nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24863(methyl({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d...)
Affinity DataIC50: 1.52E+3nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24859(({4-[2-(methylsulfanyl)-6-phenylpyrido[2,3-d]pyrim...)
Affinity DataIC50: 1.71E+3nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
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