Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50022383
TargetBeta-secretase 1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50182869(N-((S)-2-amino-3-((S)-1-((S)-1-((2S,3R)-4-(3,5-di(...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human recombinant BACE1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50157441(5-{(S)-3-[2-((S)-2-{(2S,3S)-2-Amino-3-[(1H-tetrazo...)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of human recombinant BACE1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50182871(N-((2S,5S)-5-((S)-1-((1R,2S)-1-(3-(2H-Tetrazol-5-y...)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of human recombinant BACE1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50157439(3-((2R,3S)-3-((S)-2-((S)-2-((S)-2-amino-3-(2H-tetr...)
Affinity DataIC50: 8.20nMAssay Description:Inhibition of human recombinant BACE1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM16034(N-[(1S,2R)-1-benzyl-3-(cyclopropylamino)-2-hydroxy...)
Affinity DataIC50: 15nMAssay Description:Inhibition of human recombinant BACE1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM15790(CHEMBL42908 | Hydroxyethylene-Based Peptidomimetic...)
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant BACE1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50234644(N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)phenylamino)-3-h...)
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant BACE1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50234646(2-(((2S,3S)-4-(3-(2H-tetrazol-5-yl)phenylamino)-3-...)
Affinity DataIC50: 96nMAssay Description:Inhibition of human recombinant BACE1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50234643(N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)phenylamino)-3-h...)
Affinity DataIC50: 140nMAssay Description:Inhibition of human recombinant BACE1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50234645(N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)phenylamino)-3-h...)
Affinity DataIC50: 360nMAssay Description:Inhibition of human recombinant BACE1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed