Compile Data Set for Download or QSAR
maximum 50k data
Found 50 Enz. Inhib. hit(s) with all data for entry = 50038181
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24882(7-{4-[(4-{4-amino-1H-pyrazolo[3,4-d]pyrimidin-1-yl...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human recombinant Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24881(7-(4-{[4-(6-fluoro-1H-1,3-benzodiazol-2-yl)piperid...)
Affinity DataIC50:  18nMAssay Description:Inhibition of human recombinant Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372787(CHEMBL255348)
Affinity DataIC50:  21nMAssay Description:Inhibition of human recombinant Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372781(CHEMBL255835)
Affinity DataIC50:  21nMAssay Description:Inhibition of human recombinant Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM15169(1-{1-[(4-{7-phenyl-1H-imidazo[4,5-g]quinoxalin-6-y...)
Affinity DataIC50:  58nMAssay Description:Inhibition of human recombinant Akt1More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372782(CHEMBL402579)
Affinity DataIC50:  69nMAssay Description:Inhibition of human recombinant Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372784(CHEMBL402199)
Affinity DataIC50:  81nMAssay Description:Inhibition of human recombinant Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372781(CHEMBL255835)
Affinity DataIC50:  85nMAssay Description:Inhibition of human recombinant Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372790(CHEMBL270157)
Affinity DataIC50:  86nMAssay Description:Inhibition of human recombinant Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24882(7-{4-[(4-{4-amino-1H-pyrazolo[3,4-d]pyrimidin-1-yl...)
Affinity DataIC50:  99nMAssay Description:Inhibition of human recombinant Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372785(CHEMBL401999)
Affinity DataIC50:  107nMAssay Description:Inhibition of human recombinant Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372789(CHEMBL401622)
Affinity DataIC50:  121nMAssay Description:Inhibition of human recombinant Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372783(CHEMBL255360)
Affinity DataIC50:  129nMAssay Description:Inhibition of human recombinant Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372788(CHEMBL255559)
Affinity DataIC50:  131nMAssay Description:Inhibition of human recombinant Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM15169(1-{1-[(4-{7-phenyl-1H-imidazo[4,5-g]quinoxalin-6-y...)
Affinity DataIC50:  210nMAssay Description:Inhibition of human recombinant Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372782(CHEMBL402579)
Affinity DataIC50:  221nMAssay Description:Inhibition of Akt1 phosphorylation in human C33a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24881(7-(4-{[4-(6-fluoro-1H-1,3-benzodiazol-2-yl)piperid...)
Affinity DataIC50:  239nMAssay Description:Inhibition of human recombinant Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372786(CHEMBL270815)
Affinity DataIC50:  244nMAssay Description:Inhibition of human recombinant Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372795(CHEMBL270388)
Affinity DataIC50:  253nMAssay Description:Inhibition of human recombinant Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372784(CHEMBL402199)
Affinity DataIC50:  259nMAssay Description:Inhibition of human recombinant Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372785(CHEMBL401999)
Affinity DataIC50:  274nMAssay Description:Inhibition of human recombinant Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24881(7-(4-{[4-(6-fluoro-1H-1,3-benzodiazol-2-yl)piperid...)
Affinity DataIC50:  277nMAssay Description:Inhibition of Akt1 phosphorylation in human C33a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372782(CHEMBL402579)
Affinity DataIC50:  281nMAssay Description:Inhibition of human recombinant Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24882(7-{4-[(4-{4-amino-1H-pyrazolo[3,4-d]pyrimidin-1-yl...)
Affinity DataIC50:  295nMAssay Description:Inhibition of Akt1 phosphorylation in human C33a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372782(CHEMBL402579)
Affinity DataIC50:  344nMAssay Description:Inhibition of Akt2 phosphorylation in human C33a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372781(CHEMBL255835)
Affinity DataIC50:  463nMAssay Description:Inhibition of Akt1 phosphorylation in human C33a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24882(7-{4-[(4-{4-amino-1H-pyrazolo[3,4-d]pyrimidin-1-yl...)
Affinity DataIC50:  468nMAssay Description:Inhibition of Akt2 phosphorylation in human C33a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372794(CHEMBL429576)
Affinity DataIC50:  495nMAssay Description:Inhibition of human recombinant Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372789(CHEMBL401622)
Affinity DataIC50:  556nMAssay Description:Inhibition of human recombinant Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372786(CHEMBL270815)
Affinity DataIC50:  577nMAssay Description:Inhibition of human recombinant Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372783(CHEMBL255360)
Affinity DataIC50:  696nMAssay Description:Inhibition of human recombinant Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372787(CHEMBL255348)
Affinity DataIC50:  839nMAssay Description:Inhibition of human recombinant Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372781(CHEMBL255835)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Akt2 phosphorylation in human C33a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372788(CHEMBL255559)
Affinity DataIC50:  1.23E+3nMAssay Description:Inhibition of human recombinant Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24881(7-(4-{[4-(6-fluoro-1H-1,3-benzodiazol-2-yl)piperid...)
Affinity DataIC50:  1.81E+3nMAssay Description:Inhibition of Akt2 phosphorylation in human C33a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372784(CHEMBL402199)
Affinity DataIC50:  1.83E+3nMAssay Description:Inhibition of Akt1 phosphorylation in human C33a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372794(CHEMBL429576)
Affinity DataIC50:  2.06E+3nMAssay Description:Inhibition of human recombinant Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM15169(1-{1-[(4-{7-phenyl-1H-imidazo[4,5-g]quinoxalin-6-y...)
Affinity DataIC50: >2.12E+3nMAssay Description:Inhibition of human recombinant Akt3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372793(CHEMBL255772)
Affinity DataIC50:  2.25E+3nMAssay Description:Inhibition of human recombinant Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM15148(2,3-diphenylquinoxaline 1 | 2-[4-(3-phenylquinoxal...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of human recombinant Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372784(CHEMBL402199)
Affinity DataIC50:  5.08E+3nMAssay Description:Inhibition of Akt2 phosphorylation in human C33a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372791(CHEMBL402355)
Affinity DataIC50:  5.55E+3nMAssay Description:Inhibition of human recombinant Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372795(CHEMBL270388)
Affinity DataIC50:  7.36E+3nMAssay Description:Inhibition of human recombinant Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372790(CHEMBL270157)
Affinity DataIC50:  7.36E+3nMAssay Description:Inhibition of human recombinant Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372793(CHEMBL255772)
Affinity DataIC50:  8.14E+3nMAssay Description:Inhibition of human recombinant Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372792(CHEMBL257441)
Affinity DataIC50:  8.46E+3nMAssay Description:Inhibition of human recombinant Akt1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372792(CHEMBL257441)
Affinity DataIC50:  1.54E+4nMAssay Description:Inhibition of human recombinant Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM15148(2,3-diphenylquinoxaline 1 | 2-[4-(3-phenylquinoxal...)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of human recombinant Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50372791(CHEMBL402355)
Affinity DataIC50:  3.77E+4nMAssay Description:Inhibition of human recombinant Akt2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM15148(2,3-diphenylquinoxaline 1 | 2-[4-(3-phenylquinoxal...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant Akt3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed