Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50025815
TargetGlucocorticoid receptor(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50247195((8S,9R,10S,11S,13S,14S,16R,17R)-N-(2-(2-(2-(((3S,5...)
Affinity DataEC50:  33nMAssay Description:Transcriptional activation of Gal4(1-147) tagged glucocorticoid receptor in human HeLa cells by luciferase reporter gene assay relative to OxDex-AEEAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50247196((8S,9R,10S,11S,13S,14S,16R,17R)-N-((2R,5R,8R)-1-am...)
Affinity DataEC50:  1.86E+3nMAssay Description:Transcriptional activation of Gal4(1-147) tagged glucocorticoid receptor in human HeLa cells by luciferase reporter gene assay relative to OxDex-AEEAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50247194(9-Fluoro-11,17-dihydroxy-10,13,16-trimethyl-3-oxo-...)
Affinity DataEC50:  2.50E+3nMAssay Description:Transcriptional activation of Gal4(1-147) tagged glucocorticoid receptor in human HeLa cells by luciferase reporter gene assay relative to OxDex-AEEAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed