Compile Data Set for Download or QSAR
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Found 7 Enz. Inhib. hit(s) with all data for entry = 50038566
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50261457(17-(Cyclopropylmethyl)-4,6alpha-epoxymethanomorphi...)
Affinity DataIC50:  0.980nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataIC50:  1.14nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50261457(17-(Cyclopropylmethyl)-4,6alpha-epoxymethanomorphi...)
Affinity DataIC50:  1.21nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in ICR mouse whole brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataIC50:  1.27nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in ICR mouse whole brainMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50039029((+)-4-((alpha R)-((2S,5R)-4-allyl-2,5-dimethylpipe...)
Affinity DataIC50:  6.41nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in ICR mouse whole brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50261457(17-(Cyclopropylmethyl)-4,6alpha-epoxymethanomorphi...)
Affinity DataIC50:  57.3nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in ICR mouse whole brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50261458(4,6alpha-Epoxymethano-3-methoxy-17-methylmorphinan...)
Affinity DataIC50:  183nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in ICR mouse whole brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed