Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50038449
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50376590(CHEMBL402207)
Affinity DataIC50: >1.00E+3nMAssay Description:Antagonist activity at human muscarinic M4 receptor expressed in CHO cells assessed as blockade of carbachol-induced inhibition of forskolin-stimulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50071171(9-Methoxy-2-methyl-11,12-dihydro-3H,6aH,13H-6-oxa-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Antagonist activity at human muscarinic M4 receptor expressed in CHO cells assessed as blockade of carbachol-induced inhibition of forskolin-stimulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50376591(CHEMBL403773)
Affinity DataEC50:  138nMAssay Description:Antagonist activity at human muscarinic M4 receptor expressed in CHO cells assessed as blockade of carbachol-induced inhibition of forskolin-stimulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50071171(9-Methoxy-2-methyl-11,12-dihydro-3H,6aH,13H-6-oxa-...)
Affinity DataEC50:  54nMAssay Description:Antagonist activity at human muscarinic M4 receptor expressed in CHO cells assessed as blockade of carbachol-induced inhibition of forskolin-stimulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50376590(CHEMBL402207)
Affinity DataEC50:  67nMAssay Description:Antagonist activity at human muscarinic M4 receptor expressed in CHO cells assessed as blockade of carbachol-induced inhibition of forskolin-stimulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed