Affinity DataIC50: 631nMAssay Description:Inhibition of human recombinant urotensin 2 receptor-mediated calcium mobilization expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataKd: 10nMAssay Description:Antagonist activity at human urotensin 2 receptorMore data for this Ligand-Target Pair