Compile Data Set for Download or QSAR
Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 2775
LigandChemical structure of BindingDB Monomer ID 24496BDBM24496(3-(3-fluoro-4-{[2-(pyrrolidin-1-ylcarbonyl)thieno[...)
Affinity DataIC50: 9nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24498BDBM24498(CHEMBL254760 | 3-(3-fluoro-4-{[2-(1-methyl-1H-imid...)
Affinity DataIC50: 10nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24500BDBM24500(3-(3-fluoro-4-{[2-(1-methyl-1H-imidazol-2-yl)thien...)
Affinity DataIC50: 10nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24499BDBM24499(3-(4-{[2-(1-ethyl-1H-imidazol-4-yl)thieno[3,2-b]py...)
Affinity DataIC50: 11nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24505BDBM24505(3-(3-fluoro-4-{[2-(pyridin-2-yl)thieno[3,2-b]pyrid...)
Affinity DataIC50: 17nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24504BDBM24504(3-(3-fluoro-4-{[2-(1,3-thiazol-2-yl)thieno[3,2-b]p...)
Affinity DataIC50: 17nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24493BDBM24493(7-(2-fluoro-4-{[(1-phenylacetamido)methanethioyl]a...)
Affinity DataIC50: 19nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24502BDBM24502(3-(3-fluoro-4-{[2-(1-methyl-1H-pyrazol-4-yl)thieno...)
Affinity DataIC50: 24nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24501BDBM24501(3-(4-{[2-(1-ethyl-1H-imidazol-2-yl)thieno[3,2-b]py...)
Affinity DataIC50: 25nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24502BDBM24502(3-(3-fluoro-4-{[2-(1-methyl-1H-pyrazol-4-yl)thieno...)
Affinity DataIC50: 25nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24503BDBM24503(3-(3-fluoro-4-{[2-(1-methyl-1H-1,2,4-triazol-5-yl)...)
Affinity DataIC50: 28nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24498BDBM24498(CHEMBL254760 | 3-(3-fluoro-4-{[2-(1-methyl-1H-imid...)
Affinity DataIC50: 29nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24510BDBM24510(3-(3-fluoro-4-{[2-(1-methyl-1H-pyrrol-2-yl)thieno[...)
Affinity DataIC50: 31nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24509BDBM24509(3-(3-fluoro-4-{[2-(thiophen-2-yl)thieno[3,2-b]pyri...)
Affinity DataIC50: 32nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24485BDBM24485(3-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophe...)
Affinity DataIC50: 32nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24493BDBM24493(7-(2-fluoro-4-{[(1-phenylacetamido)methanethioyl]a...)
Affinity DataIC50: 48nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24510BDBM24510(3-(3-fluoro-4-{[2-(1-methyl-1H-pyrrol-2-yl)thieno[...)
Affinity DataIC50: 49nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24500BDBM24500(3-(3-fluoro-4-{[2-(1-methyl-1H-imidazol-2-yl)thien...)
Affinity DataIC50: 51nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24499BDBM24499(3-(4-{[2-(1-ethyl-1H-imidazol-4-yl)thieno[3,2-b]py...)
Affinity DataIC50: 52nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24496BDBM24496(3-(3-fluoro-4-{[2-(pyrrolidin-1-ylcarbonyl)thieno[...)
Affinity DataIC50: 54nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24508BDBM24508(3-(3-fluoro-4-{[2-(1,3,4-thiadiazol-2-yl)thieno[3,...)
Affinity DataIC50: 60nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24505BDBM24505(3-(3-fluoro-4-{[2-(pyridin-2-yl)thieno[3,2-b]pyrid...)
Affinity DataIC50: 62nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24512BDBM24512(3-(3-fluoro-4-{[2-(pyrimidin-5-yl)thieno[3,2-b]pyr...)
Affinity DataIC50: 63nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24504BDBM24504(3-(3-fluoro-4-{[2-(1,3-thiazol-2-yl)thieno[3,2-b]p...)
Affinity DataIC50: 65nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24491BDBM24491(7-(2-fluoro-4-{[(1-phenylacetamido)methanethioyl]a...)
Affinity DataIC50: 65nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24503BDBM24503(3-(3-fluoro-4-{[2-(1-methyl-1H-1,2,4-triazol-5-yl)...)
Affinity DataIC50: 69nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24509BDBM24509(3-(3-fluoro-4-{[2-(thiophen-2-yl)thieno[3,2-b]pyri...)
Affinity DataIC50: 70nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24511BDBM24511(3-(3-fluoro-4-{[2-(furan-3-yl)thieno[3,2-b]pyridin...)
Affinity DataIC50: 74nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24492BDBM24492(7-(2-fluoro-4-{[(1-phenylacetamido)methanethioyl]a...)
Affinity DataIC50: 80nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24490BDBM24490(methyl 7-(2-fluoro-4-{[(1-phenylacetamido)methanet...)
Affinity DataIC50: 90nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24507BDBM24507(3-(3-fluoro-4-{[2-(pyrimidin-2-yl)thieno[3,2-b]pyr...)
Affinity DataIC50: 94nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24501BDBM24501(3-(4-{[2-(1-ethyl-1H-imidazol-2-yl)thieno[3,2-b]py...)
Affinity DataIC50: 108nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24506BDBM24506(3-(3-fluoro-4-{[2-(pyridin-3-yl)thieno[3,2-b]pyrid...)
Affinity DataIC50: 113nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24490BDBM24490(methyl 7-(2-fluoro-4-{[(1-phenylacetamido)methanet...)
Affinity DataIC50: 113nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24494BDBM24494(N,N-diethyl-7-(2-fluoro-4-{[(1-phenylacetamido)met...)
Affinity DataIC50: 114nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24486BDBM24486(3-(3-fluoro-4-{thieno[3,2-b]pyridin-7-yloxy}phenyl...)
Affinity DataIC50: 116nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24485BDBM24485(3-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophe...)
Affinity DataIC50: 121nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24495BDBM24495(3-(3-fluoro-4-{[2-(morpholin-4-ylcarbonyl)thieno[3...)
Affinity DataIC50: 125nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24506BDBM24506(3-(3-fluoro-4-{[2-(pyridin-3-yl)thieno[3,2-b]pyrid...)
Affinity DataIC50: 126nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24489BDBM24489(3-(3-fluoro-4-{[2-(furan-2-ylcarbonyl)thieno[3,2-b...)
Affinity DataIC50: 127nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24491BDBM24491(7-(2-fluoro-4-{[(1-phenylacetamido)methanethioyl]a...)
Affinity DataIC50: 129nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24488BDBM24488(3-(3-fluoro-4-{[2-(methylsulfanyl)thieno[3,2-b]pyr...)
Affinity DataIC50: 130nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24489BDBM24489(3-(3-fluoro-4-{[2-(furan-2-ylcarbonyl)thieno[3,2-b...)
Affinity DataIC50: 130nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24487BDBM24487(CHEMBL256715 | 3-(3-fluoro-4-{[2-(1-hydroxyethyl)t...)
Affinity DataIC50: 132nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24492BDBM24492(7-(2-fluoro-4-{[(1-phenylacetamido)methanethioyl]a...)
Affinity DataIC50: 133nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24508BDBM24508(3-(3-fluoro-4-{[2-(1,3,4-thiadiazol-2-yl)thieno[3,...)
Affinity DataIC50: 145nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24512BDBM24512(3-(3-fluoro-4-{[2-(pyrimidin-5-yl)thieno[3,2-b]pyr...)
Affinity DataIC50: 175nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24507BDBM24507(3-(3-fluoro-4-{[2-(pyrimidin-2-yl)thieno[3,2-b]pyr...)
Affinity DataIC50: 181nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Methylgene

LigandChemical structure of BindingDB Monomer ID 24497BDBM24497(3-[3-fluoro-4-({2-[(4-methylpiperazin-1-yl)carbony...)
Affinity DataIC50: 193nMpH: 7.5 T: 2°CAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24495BDBM24495(3-(3-fluoro-4-{[2-(morpholin-4-ylcarbonyl)thieno[3...)
Affinity DataIC50: 289nMAssay Description:Inhibition of kinase activity was measured in a DELFIA assay (Perkin-Elmer). The substrate poly (Glu4, Tyr) was immobilized onto black high-binding p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2008
Entry Details Article
PubMed
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