Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50026025
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260622((S)-7-(Toluene-4-sulfonyl)-1,4-dioxa-7-aza-spiro[4...)
Affinity DataIC50: 3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260661((S)-2-(Toluene-4-sulfonyl)-6,10-dioxa-2-aza-spiro-...)
Affinity DataIC50: 6nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260662((S)-2-(Toluene-4-sulfonyl)-6,11-dioxa-2-aza-spiro-...)
Affinity DataIC50: 8nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260663((S)-7-Benzenesulfonyl-1,4-dioxa-7-aza-spiro[4.4]-n...)
Affinity DataIC50: 8nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247539(N-((3S,5S)-1-((E)-3-(3,4-dimethoxyphenyl)acryloyl)...)
Affinity DataIC50: 9nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260664((S)-2-Benzenesulfonyl-6,10-dioxa-2-aza-spiro[4.5]-...)
Affinity DataIC50: 11nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260665((S)-2-Benzenesulfonyl-6,11-dioxa-2-aza-spiro[4.6]-...)
Affinity DataIC50: 12nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50253922(trans-4-Hydroxy-1-(toluene-4-sulfonyl)-pyrrolidine...)
Affinity DataIC50: 100nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260537((S)-7-(Toluene-4-sulfonyl)-1,4-dioxa-7-aza-spiro[4...)
Affinity DataIC50: 100nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260619((S)-7-Benzenesulfonyl-1,4-dioxa-7-aza-spiro[4.4]no...)
Affinity DataIC50: 200nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260617((S)-2-(Toluene-4-sulfonyl)-6,10-dioxa-2-aza-spiro[...)
Affinity DataIC50: 200nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260618((S)-2-(Toluene-4-sulfonyl)-6,11-dioxa-2-aza-spiro-...)
Affinity DataIC50: 300nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260507(4-Oxo-1-(toluene-4-sulfonyl)-pyrrolidine-2-carboxy...)
Affinity DataIC50: 400nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50253923(1-Benzenesulfonyl-4-hydroxy-pyrrolidine-2-carboxyl...)
Affinity DataIC50: 800nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260620((S)-2-Benzenesulfonyl-6,10-dioxa-2-aza-spiro-[4.5]...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260621((S)-2-Benzenesulfonyl-6,11-dioxa-2-aza-spiro[4.6]-...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260508(1-Benzenesulfonyl-4-oxo-pyrrolidine-2-carboxylicac...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50253924(trans-4-Hydroxy-1-methanesulfonyl-pyrrolidine-2-ca...)
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260509(1-Methanesulfonyl-4-oxo-pyrrolidine-2-carboxylicac...)
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50253922(trans-4-Hydroxy-1-(toluene-4-sulfonyl)-pyrrolidine...)
Affinity DataIC50: 3.84E+4nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50253924(trans-4-Hydroxy-1-methanesulfonyl-pyrrolidine-2-ca...)
Affinity DataIC50: 4.16E+4nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260622((S)-7-(Toluene-4-sulfonyl)-1,4-dioxa-7-aza-spiro[4...)
Affinity DataIC50: 4.85E+4nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50253923(1-Benzenesulfonyl-4-hydroxy-pyrrolidine-2-carboxyl...)
Affinity DataIC50: 5.38E+4nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260507(4-Oxo-1-(toluene-4-sulfonyl)-pyrrolidine-2-carboxy...)
Affinity DataIC50: 5.49E+4nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260663((S)-7-Benzenesulfonyl-1,4-dioxa-7-aza-spiro[4.4]-n...)
Affinity DataIC50: 5.78E+4nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260661((S)-2-(Toluene-4-sulfonyl)-6,10-dioxa-2-aza-spiro-...)
Affinity DataIC50: 6.18E+4nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260662((S)-2-(Toluene-4-sulfonyl)-6,11-dioxa-2-aza-spiro-...)
Affinity DataIC50: 7.32E+4nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260508(1-Benzenesulfonyl-4-oxo-pyrrolidine-2-carboxylicac...)
Affinity DataIC50: 7.58E+4nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260664((S)-2-Benzenesulfonyl-6,10-dioxa-2-aza-spiro[4.5]-...)
Affinity DataIC50: 8.27E+4nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260509(1-Methanesulfonyl-4-oxo-pyrrolidine-2-carboxylicac...)
Affinity DataIC50: 9.26E+4nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260665((S)-2-Benzenesulfonyl-6,11-dioxa-2-aza-spiro[4.6]-...)
Affinity DataIC50: 1.07E+5nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260618((S)-2-(Toluene-4-sulfonyl)-6,11-dioxa-2-aza-spiro-...)
Affinity DataIC50: 1.24E+5nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260621((S)-2-Benzenesulfonyl-6,11-dioxa-2-aza-spiro[4.6]-...)
Affinity DataIC50: 1.35E+5nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50247539(N-((3S,5S)-1-((E)-3-(3,4-dimethoxyphenyl)acryloyl)...)
Affinity DataIC50: 1.42E+5nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260619((S)-7-Benzenesulfonyl-1,4-dioxa-7-aza-spiro[4.4]no...)
Affinity DataIC50: 1.51E+5nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260537((S)-7-(Toluene-4-sulfonyl)-1,4-dioxa-7-aza-spiro[4...)
Affinity DataIC50: 1.56E+5nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260620((S)-2-Benzenesulfonyl-6,10-dioxa-2-aza-spiro-[4.5]...)
Affinity DataIC50: 1.68E+5nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50260617((S)-2-(Toluene-4-sulfonyl)-6,10-dioxa-2-aza-spiro[...)
Affinity DataIC50: 1.74E+5nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed