Compile Data Set for Download or QSAR
maximum 50k data
Found 36 Enz. Inhib. hit(s) with all data for entry = 50026283
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244360((6aR,10aR)-6,6,9-trimethyl-3-(2-(thiophen-2-yl)pro...)
Affinity DataKi:  0.270nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244359((6aR,10aR)-3-(2-(3-bromophenyl)propan-2-yl)-6,6,9-...)
Affinity DataKi:  0.540nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244284((6aR,10aR)-3-(2-(4-ethylphenyl)propan-2-yl)-6,6,9-...)
Affinity DataKi:  0.670nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244252((6aR,10aR)-6,6,9-trimethyl-3-(2-p-tolylpropan-2-yl...)
Affinity DataKi:  0.880nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244322((6aR,10aR)-3-(2-(3-fluorophenyl)propan-2-yl)-6,6,9...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50133546((6aR,10aR)-6,6,9-Trimethyl-3-(1-methyl-1-phenyl-et...)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50243718(3-(2-((6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10...)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244360((6aR,10aR)-6,6,9-trimethyl-3-(2-(thiophen-2-yl)pro...)
Affinity DataKi:  1.08nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244281((6aR,10aR)-6,6,9-trimethyl-3-(2-m-tolylpropan-2-yl...)
Affinity DataKi:  1.13nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244358((6aR,10aR)-3-(2-(4-bromophenyl)propan-2-yl)-6,6,9-...)
Affinity DataKi:  1.54nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244359((6aR,10aR)-3-(2-(3-bromophenyl)propan-2-yl)-6,6,9-...)
Affinity DataKi:  1.59nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244323((6aR,10aR)-3-(2-(4-chlorophenyl)propan-2-yl)-6,6,9...)
Affinity DataKi:  1.68nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244320((6aR,10aR)-6,6,9-trimethyl-3-(2-(4-propylphenyl)pr...)
Affinity DataKi:  1.77nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244284((6aR,10aR)-3-(2-(4-ethylphenyl)propan-2-yl)-6,6,9-...)
Affinity DataKi:  1.85nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244281((6aR,10aR)-6,6,9-trimethyl-3-(2-m-tolylpropan-2-yl...)
Affinity DataKi:  2.53nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50243717(3-[1-(4-Cyano-phenyl)-1-methyl-ethyl]-6,6,9-trimet...)
Affinity DataKi:  2.53nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50243718(3-(2-((6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10...)
Affinity DataKi:  2.72nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244357((6aR,10aR)-3-(2-(3-chlorophenyl)propan-2-yl)-6,6,9...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244252((6aR,10aR)-6,6,9-trimethyl-3-(2-p-tolylpropan-2-yl...)
Affinity DataKi:  3.13nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244357((6aR,10aR)-3-(2-(3-chlorophenyl)propan-2-yl)-6,6,9...)
Affinity DataKi:  3.54nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244358((6aR,10aR)-3-(2-(4-bromophenyl)propan-2-yl)-6,6,9-...)
Affinity DataKi:  5.03nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244322((6aR,10aR)-3-(2-(3-fluorophenyl)propan-2-yl)-6,6,9...)
Affinity DataKi:  5.26nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244283((6aR,10aR)-3-(2-(3,5-dimethylphenyl)propan-2-yl)-6...)
Affinity DataKi:  7.45nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244320((6aR,10aR)-6,6,9-trimethyl-3-(2-(4-propylphenyl)pr...)
Affinity DataKi:  7.83nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50243717(3-[1-(4-Cyano-phenyl)-1-methyl-ethyl]-6,6,9-trimet...)
Affinity DataKi:  9.25nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244282((6aR,10aR)-6,6,9-trimethyl-3-(2-o-tolylpropan-2-yl...)
Affinity DataKi:  10.7nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244283((6aR,10aR)-3-(2-(3,5-dimethylphenyl)propan-2-yl)-6...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50133546((6aR,10aR)-6,6,9-Trimethyl-3-(1-methyl-1-phenyl-et...)
Affinity DataKi:  12.3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244321((6aR,10aR)-3-(2-(4-fluorophenyl)propan-2-yl)-6,6,9...)
Affinity DataKi:  12.4nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50243719(CHEMBL471367 | N-{3-[1-(1-hydroxy-6,6,9-trimethyl)...)
Affinity DataKi:  13.6nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50243719(CHEMBL471367 | N-{3-[1-(1-hydroxy-6,6,9-trimethyl)...)
Affinity DataKi:  13.7nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244323((6aR,10aR)-3-(2-(4-chlorophenyl)propan-2-yl)-6,6,9...)
Affinity DataKi:  18.8nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50067734((-)-(6aR-trans)-6,6,9-trimethyl-3-pentyl-6a,7,10,1...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50067734((-)-(6aR-trans)-6,6,9-trimethyl-3-pentyl-6a,7,10,1...)
Affinity DataKi:  28.5nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244282((6aR,10aR)-6,6,9-trimethyl-3-(2-o-tolylpropan-2-yl...)
Affinity DataKi:  34.4nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244321((6aR,10aR)-3-(2-(4-fluorophenyl)propan-2-yl)-6,6,9...)
Affinity DataKi:  76.1nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed