Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50026408
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50252375(CHEMBL446072 | Spheciosterol sulfate C)
Affinity DataIC50:  110nMAssay Description:Inhibition of PKCzeta (unknown origin) by TR-FRET based lanthascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50252374(CHEMBL475118 | Spheciosterol sulfate B)
Affinity DataIC50:  530nMAssay Description:Inhibition of PKCzeta (unknown origin) by TR-FRET based lanthascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50252376(CHEMBL455091 | Topsentiasterol sulfate E)
Affinity DataIC50:  1.21E+3nMAssay Description:Inhibition of PKCzeta (unknown origin) by TR-FRET based lanthascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50252373(CHEMBL447723 | Spheciosterol sulfate A)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of PKCzeta (unknown origin) by TR-FRET based lanthascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor p65(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50252374(CHEMBL475118 | Spheciosterol sulfate B)
Affinity DataEC50:  1.20E+4nMAssay Description:Inhibition of IL1-induced NFkappaB P65 activation in human osteoarthritic primary chondrocytes preincubated 2 hrs before addition of IL1 by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor p65(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50252375(CHEMBL446072 | Spheciosterol sulfate C)
Affinity DataEC50:  1.20E+4nMAssay Description:Inhibition of IL1-induced NFkappaB P65 activation in human osteoarthritic primary chondrocytes preincubated 2 hrs before addition of IL1 by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor p65(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50252373(CHEMBL447723 | Spheciosterol sulfate A)
Affinity DataEC50:  1.20E+4nMAssay Description:Inhibition of IL1-induced NFkappaB P65 activation in human osteoarthritic primary chondrocytes preincubated 2 hrs before addition of IL1 by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor p65(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50252376(CHEMBL455091 | Topsentiasterol sulfate E)
Affinity DataEC50:  1.20E+4nMAssay Description:Inhibition of IL1-induced NFkappaB P65 activation in human osteoarthritic primary chondrocytes preincubated 2 hrs before addition of IL1 by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed