Report error Found 65 Enz. Inhib. hit(s) with all data for entry = 50026566
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 8.20nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 10.7nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 32.4nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 167nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 321nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 474nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 542nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 572nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:Antagonist activity at human cloned 5HT2C receptor expressed in CHO cell assessed as blockade of 5-HT-stimulated [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 667nMAssay Description:Displacement of [3H]LSD from human cloned 5HT6 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]LSD from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D4 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D3 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 2.25E+3nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 6.37E+3nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 9.44E+3nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]LSD from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]LSD from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]LSD from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]LSD from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]LSD from human cloned 5HT6 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]LSD from human cloned 5HT6 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]LSD from human cloned 5HT6 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]LSD from human cloned 5HT6 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Human)
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Korea Research Institute of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT1A receptorMore data for this Ligand-Target Pair





















