Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50026705
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50273238((S,S)-beta-3 Fluoro-Benzylaspartate | CHEMBL457411)
Affinity DataIC50:  2.46E+3nMAssay Description:Displacement of [3H]D-aspartate from human EAAT3 expressed in mouse C17.2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50273197(CHEMBL455918 | L-threo-beta-(1-naphthyl)methyloxas...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of [14C]glutamate uptake at human EAAT3 expressed in african green monkey COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50273237(CHEMBL458065 | L-threo-beta-(2-naphthyl)methyloxas...)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of [14C]glutamate uptake at human EAAT3 expressed in african green monkey COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50093753((2S,3S)-2-Amino-3-benzyloxy-succinic acid | (2S,3S...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of [14C]glutamate uptake at human EAAT3 expressed in african green monkey COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50273239((S,R)-beta-3 Fluoro-Benzylaspartate | CHEMBL457412)
Affinity DataIC50:  2.11E+4nMAssay Description:Displacement of [3H]D-aspartate from human EAAT3 expressed in mouse C17.2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed