Compile Data Set for Download or QSAR
Report error Found 105 Enz. Inhib. hit(s) with all data for entry = 3143
LigandChemical structure of BindingDB Monomer ID 28674BDBM28674(2-({3-[(2-carboxy-4-chlorophenyl)carbamoyl]benzene...)
Affinity DataIC50: 4nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28691BDBM28691(5-methyl-2-({3-[(7-methyl-1H-indole-1-)sulfonyl]be...)
Affinity DataIC50: 4nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28661BDBM28661(GW501516 | CHEMBL38943 | 2-{2-methyl-4-[({4-methyl...)
Affinity DataIC50: 5nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28669BDBM28669(2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)b...)
Affinity DataIC50: 5nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28670BDBM28670(4-bromo-2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-su...)
Affinity DataIC50: 5nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28695BDBM28695(5-chloro-2-({3-[(4-methoxy-1H-indole-1-)sulfonyl]b...)
Affinity DataIC50: 6nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28682BDBM28682(5-methyl-2-({3-[(4-methyl-1H-indole-1-)sulfonyl]be...)
Affinity DataIC50: 6nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28666BDBM28666(5-chloro-2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-s...)
Affinity DataIC50: 8nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28667BDBM28667(5-bromo-2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-su...)
Affinity DataIC50: 8nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28688BDBM28688(5-methyl-2-({3-[(6-methyl-1H-indole-1-)sulfonyl]be...)
Affinity DataIC50: 10nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28675BDBM28675(2-[(3-{[5-(carboxymethoxy)-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50: 10nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28676BDBM28676(5-chloro-2-({3-[(6-methoxy-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50: 10nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28683BDBM28683(2-({3-[(4-bromo-1H-indole-1-)sulfonyl]benzene}amid...)
Affinity DataIC50: 10nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28684BDBM28684(2-({3-[(4-methoxy-1H-indole-1-)sulfonyl]benzene}am...)
Affinity DataIC50: 10nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28685BDBM28685(5-methyl-2-({3-[(5-methyl-1H-indole-1-)sulfonyl]be...)
Affinity DataIC50: 10nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28672BDBM28672(5-chloro-2-({3-[(5-methoxy-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50: 13nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28665BDBM28665(5-methyl-2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-s...)
Affinity DataIC50: 13nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28696BDBM28696(5-chloro-2-({3-[(5-methoxy-1H-indole-1-)sulfonyl]b...)
Affinity DataIC50: 13nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28697BDBM28697(5-chloro-2-({3-[(6-methoxy-1H-indole-1-)sulfonyl]b...)
Affinity DataIC50: 13nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28677BDBM28677(5-chloro-2-({3-[(7-fluoro-1,2,3,4-tetrahydroisoqui...)
Affinity DataIC50: 16nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28692BDBM28692(2-({3-[(7-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50: 16nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28679BDBM28679(5-chloro-2-({3-[(7-chloro-8-methyl-1,2,3,4-tetrahy...)
Affinity DataIC50: 16nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28698BDBM28698(5-chloro-2-({3-[(5-methoxy-4-methyl-1H-indole-1-)s...)
Affinity DataIC50: 16nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28686BDBM28686(2-({3-[(5-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50: 20nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28673BDBM28673(5-chloro-2-({3-[(5-hydroxy-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50: 20nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28694BDBM28694(2-({3-[(5-methoxy-4-methyl-1H-indole-1-)sulfonyl]b...)
Affinity DataIC50: 20nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28678BDBM28678(5-chloro-2-({3-[(7-chloro-1,2,3,4-tetrahydroisoqui...)
Affinity DataIC50: 25nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28668BDBM28668(5-fluoro-2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-s...)
Affinity DataIC50: 25nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28690BDBM28690(2-({3-[(6-methoxy-1H-indole-1-)sulfonyl]benzene}am...)
Affinity DataIC50: 32nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28693BDBM28693(2-({3-[(7-methoxy-1H-indole-1-)sulfonyl]benzene}am...)
Affinity DataIC50: 50nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28689BDBM28689(2-({3-[(6-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50: 63nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28663BDBM28663(2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)b...)
Affinity DataIC50: 126nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 28687BDBM28687(2-({3-[(5-methoxy-1H-indole-1-)sulfonyl]benzene}am...)
Affinity DataIC50: 158nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28692BDBM28692(2-({3-[(7-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50: 794nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28695BDBM28695(5-chloro-2-({3-[(4-methoxy-1H-indole-1-)sulfonyl]b...)
Affinity DataIC50: 794nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28685BDBM28685(5-methyl-2-({3-[(5-methyl-1H-indole-1-)sulfonyl]be...)
Affinity DataIC50: 1.00E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28691BDBM28691(5-methyl-2-({3-[(7-methyl-1H-indole-1-)sulfonyl]be...)
Affinity DataIC50: 1.00E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28682BDBM28682(5-methyl-2-({3-[(4-methyl-1H-indole-1-)sulfonyl]be...)
Affinity DataIC50: 1.00E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28683BDBM28683(2-({3-[(4-bromo-1H-indole-1-)sulfonyl]benzene}amid...)
Affinity DataIC50: 1.26E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28684BDBM28684(2-({3-[(4-methoxy-1H-indole-1-)sulfonyl]benzene}am...)
Affinity DataIC50: 1.26E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28683BDBM28683(2-({3-[(4-bromo-1H-indole-1-)sulfonyl]benzene}amid...)
Affinity DataIC50: 1.26E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28684BDBM28684(2-({3-[(4-methoxy-1H-indole-1-)sulfonyl]benzene}am...)
Affinity DataIC50: 1.59E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28686BDBM28686(2-({3-[(5-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50: 1.59E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28691BDBM28691(5-methyl-2-({3-[(7-methyl-1H-indole-1-)sulfonyl]be...)
Affinity DataIC50: 1.59E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28697BDBM28697(5-chloro-2-({3-[(6-methoxy-1H-indole-1-)sulfonyl]b...)
Affinity DataIC50: 1.59E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28669BDBM28669(2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)b...)
Affinity DataIC50: 1.59E+3nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28686BDBM28686(2-({3-[(5-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50: 2.00E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28689BDBM28689(2-({3-[(6-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50: 2.00E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28661BDBM28661(GW501516 | CHEMBL38943 | 2-{2-methyl-4-[({4-methyl...)
Affinity DataIC50: 2.00E+3nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 28695BDBM28695(5-chloro-2-({3-[(4-methoxy-1H-indole-1-)sulfonyl]b...)
Affinity DataIC50: 2.00E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
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