Compile Data Set for Download or QSAR
Report error Found 105 Enz. Inhib. hit(s) with all data for entry = 3143
LigandPNGBDBM28661(GW501516 | CHEMBL38943 | 2-{2-methyl-4-[({4-methyl...)
Affinity DataIC50: 5nM EC50:  3nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28674(2-({3-[(2-carboxy-4-chlorophenyl)carbamoyl]benzene...)
Affinity DataIC50: 4nM EC50:  1.26E+3nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28691(5-methyl-2-({3-[(7-methyl-1H-indole-1-)sulfonyl]be...)
Affinity DataIC50: 4nM EC50:  79nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28669(2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)b...)
Affinity DataIC50: 5nM EC50:  158nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28670(4-bromo-2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-su...)
Affinity DataIC50: 5nM EC50:  158nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28695(5-chloro-2-({3-[(4-methoxy-1H-indole-1-)sulfonyl]b...)
Affinity DataIC50: 6nM EC50:  158nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28682(5-methyl-2-({3-[(4-methyl-1H-indole-1-)sulfonyl]be...)
Affinity DataIC50: 6nM EC50:  20nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28666(5-chloro-2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-s...)
Affinity DataIC50: 8nM EC50:  126nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28667(5-bromo-2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-su...)
Affinity DataIC50: 8nM EC50:  200nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28688(5-methyl-2-({3-[(6-methyl-1H-indole-1-)sulfonyl]be...)
Affinity DataIC50: 10nM EC50:  50nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28675(2-[(3-{[5-(carboxymethoxy)-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50: 10nM EC50: >1.00E+4nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28676(5-chloro-2-({3-[(6-methoxy-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50: 10nM EC50:  794nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28683(2-({3-[(4-bromo-1H-indole-1-)sulfonyl]benzene}amid...)
Affinity DataIC50: 10nM EC50:  13nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28684(2-({3-[(4-methoxy-1H-indole-1-)sulfonyl]benzene}am...)
Affinity DataIC50: 10nM EC50:  40nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28685(5-methyl-2-({3-[(5-methyl-1H-indole-1-)sulfonyl]be...)
Affinity DataIC50: 10nM EC50:  32nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28672(5-chloro-2-({3-[(5-methoxy-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50: 13nM EC50:  1.26E+3nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28694(2-({3-[(5-methoxy-4-methyl-1H-indole-1-)sulfonyl]b...)
Affinity DataIC50: 20nM EC50:  13nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28665(5-methyl-2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-s...)
Affinity DataIC50: 13nM EC50:  200nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28696(5-chloro-2-({3-[(5-methoxy-1H-indole-1-)sulfonyl]b...)
Affinity DataIC50: 13nM EC50:  158nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28697(5-chloro-2-({3-[(6-methoxy-1H-indole-1-)sulfonyl]b...)
Affinity DataIC50: 13nM EC50:  100nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28677(5-chloro-2-({3-[(7-fluoro-1,2,3,4-tetrahydroisoqui...)
Affinity DataIC50: 16nM EC50:  1.00E+3nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28692(2-({3-[(7-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50: 16nM EC50:  158nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28679(5-chloro-2-({3-[(7-chloro-8-methyl-1,2,3,4-tetrahy...)
Affinity DataIC50: 16nM EC50:  316nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28698(5-chloro-2-({3-[(5-methoxy-4-methyl-1H-indole-1-)s...)
Affinity DataIC50: 16nM EC50:  16nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28686(2-({3-[(5-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50: 20nM EC50:  50nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28673(5-chloro-2-({3-[(5-hydroxy-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50: 20nM EC50:  2.00E+3nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28678(5-chloro-2-({3-[(7-chloro-1,2,3,4-tetrahydroisoqui...)
Affinity DataIC50: 25nM EC50:  794nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28668(5-fluoro-2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-s...)
Affinity DataIC50: 25nM EC50:  501nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28690(2-({3-[(6-methoxy-1H-indole-1-)sulfonyl]benzene}am...)
Affinity DataIC50: 32nM EC50:  100nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28693(2-({3-[(7-methoxy-1H-indole-1-)sulfonyl]benzene}am...)
Affinity DataIC50: 50nM EC50:  631nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28689(2-({3-[(6-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50: 63nM EC50:  200nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28663(2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)b...)
Affinity DataIC50: 126nM EC50:  1.26E+3nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM28687(2-({3-[(5-methoxy-1H-indole-1-)sulfonyl]benzene}am...)
Affinity DataIC50: 158nM EC50:  501nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28692(2-({3-[(7-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50: 794nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28695(5-chloro-2-({3-[(4-methoxy-1H-indole-1-)sulfonyl]b...)
Affinity DataIC50: 794nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28685(5-methyl-2-({3-[(5-methyl-1H-indole-1-)sulfonyl]be...)
Affinity DataIC50: 1.00E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28691(5-methyl-2-({3-[(7-methyl-1H-indole-1-)sulfonyl]be...)
Affinity DataIC50: 1.00E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28682(5-methyl-2-({3-[(4-methyl-1H-indole-1-)sulfonyl]be...)
Affinity DataIC50: 1.00E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28683(2-({3-[(4-bromo-1H-indole-1-)sulfonyl]benzene}amid...)
Affinity DataIC50: 1.26E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28684(2-({3-[(4-methoxy-1H-indole-1-)sulfonyl]benzene}am...)
Affinity DataIC50: 1.26E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28683(2-({3-[(4-bromo-1H-indole-1-)sulfonyl]benzene}amid...)
Affinity DataIC50: 1.26E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28684(2-({3-[(4-methoxy-1H-indole-1-)sulfonyl]benzene}am...)
Affinity DataIC50: 1.59E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28686(2-({3-[(5-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50: 1.59E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28691(5-methyl-2-({3-[(7-methyl-1H-indole-1-)sulfonyl]be...)
Affinity DataIC50: 1.59E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28697(5-chloro-2-({3-[(6-methoxy-1H-indole-1-)sulfonyl]b...)
Affinity DataIC50: 1.59E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28669(2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)b...)
Affinity DataIC50: 1.59E+3nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28686(2-({3-[(5-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50: 2.00E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28689(2-({3-[(6-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50: 2.00E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28661(GW501516 | CHEMBL38943 | 2-{2-methyl-4-[({4-methyl...)
Affinity DataIC50: 2.00E+3nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
LigandPNGBDBM28695(5-chloro-2-({3-[(4-methoxy-1H-indole-1-)sulfonyl]b...)
Affinity DataIC50: 2.00E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2009
Entry Details Article
PubMed
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