Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50027031
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50253820((1R,6R,9S,12S,15S,21S,24S,27S,30S,33R,36S,42S,48S,...)
Affinity DataKi:  43nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis AChBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50253821((1R,6R,9S,12S,15S,21S,24S,27S,30S,33R,36S,42S,48S,...)
Affinity DataKi:  124nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis AChBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50253825((1R,6R,9S,12S,18S,21S,24S,27S,30R,33S,39S,45S,48S,...)
Affinity DataKi:  3.10E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis AChBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50253823((1R,4S,10S,16S,19S,22R,27R,30S,33S,36S,39S,46R)-46...)
Affinity DataKi:  4.50E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis AChBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50253824((1R,6R,9S,15S,18S,21S,24S,27R,30S,36S,42S,45S,50R)...)
Affinity DataKi:  4.60E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis AChBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50253822((1R,4S,10S,16S,19S,22R,27R,30S,33S,36S,43R)-43-(2-...)
Affinity DataKi:  7.90E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from Lymnaea stagnalis AChBPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50253820((1R,6R,9S,12S,15S,21S,24S,27S,30S,33R,36S,42S,48S,...)
Affinity DataIC50:  55nMAssay Description:Activity at rat alpha7 nAChR expressed in Xenopus laevis assessed as inhibition of acetylcholine-induced current at holding potential of -80 mV by tw...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50253824((1R,6R,9S,15S,18S,21S,24S,27R,30S,36S,42S,45S,50R)...)
Affinity DataIC50:  79nMAssay Description:Activity at rat alpha7 nAChR expressed in Xenopus laevis assessed as inhibition of acetylcholine-induced current at holding potential of -80 mV by tw...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50253825((1R,6R,9S,12S,18S,21S,24S,27S,30R,33S,39S,45S,48S,...)
Affinity DataIC50:  115nMAssay Description:Activity at rat alpha7 nAChR expressed in Xenopus laevis assessed as inhibition of acetylcholine-induced current at holding potential of -80 mV by tw...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50253823((1R,4S,10S,16S,19S,22R,27R,30S,33S,36S,39S,46R)-46...)
Affinity DataIC50:  207nMAssay Description:Activity at rat alpha7 nAChR expressed in Xenopus laevis assessed as inhibition of acetylcholine-induced current at holding potential of -80 mV by tw...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50253821((1R,6R,9S,12S,15S,21S,24S,27S,30S,33R,36S,42S,48S,...)
Affinity DataIC50:  252nMAssay Description:Activity at rat alpha7 nAChR expressed in Xenopus laevis assessed as inhibition of acetylcholine-induced current at holding potential of -80 mV by tw...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50253822((1R,4S,10S,16S,19S,22R,27R,30S,33S,36S,43R)-43-(2-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Activity at rat alpha7 nAChR expressed in Xenopus laevis assessed as inhibition of acetylcholine-induced current at holding potential of -80 mV by tw...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed