Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 50022569
TargetSerine/threonine-protein kinase Chk1(Human)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50389803(CHEMBL2041933 | AZD7762)
Affinity DataKi:  3.60nMAssay Description:Binding affinity to recombinant human GST tagged Ckh1 phosphorylation expressed in baculovirus Insect cell assessed as inhibition constant incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50389803(CHEMBL2041933 | AZD7762)
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human GST tagged Ckh1 phosphorylation expressed in baculovirus Insect cell using N-biotinylaminohexanoyl-KKVSRSGLYRSPMPENLN...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed