Compile Data Set for Download or QSAR
Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50027298
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274045(3-[2-[2-(4-Cyano-phenyl)-2-oxo-ethyl]-5-(2-cyclohe...)
Affinity DataIC50: 3nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274339(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 3nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274669(N-(1-(3-(1H-imidazol-1-yl)propyl)-5-(N-methylcyclo...)
Affinity DataIC50: 4nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274340(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 4nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274471(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 4nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274470(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 4nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274246(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 5nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274671(4-cyano-N-(5-(N-methylcyclohexanecarboxamido)-1-(3...)
Affinity DataIC50: 5nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274705(4-cyano-N-(5-(N-methylcyclohexanecarboxamido)-1-(3...)
Affinity DataIC50: 5nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274558(4-cyano-N-(5-(N-methylcyclohexanecarboxamido)-1-ph...)
Affinity DataIC50: 6nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274709(N-(1-(3-amino-3-oxopropyl)-5-(N-ethylcyclohexaneca...)
Affinity DataIC50: 7nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274005(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclobutanec...)
Affinity DataIC50: 8nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274631(4-cyano-N-(1-(3-(methylamino)-3-oxopropyl)-5-(N-me...)
Affinity DataIC50: 9nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274338(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 9nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274247(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 10nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274206(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 10nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274341(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 10nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274392(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 12nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274632(4-cyano-N-(1-(3-(dimethylamino)-3-oxopropyl)-5-(N-...)
Affinity DataIC50: 14nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274629(4-cyano-N-(1-(3-methoxypropyl)-5-(N-methylcyclohex...)
Affinity DataIC50: 16nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274249(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 16nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274555(N-(1-butyl-5-(N-methylcyclohexanecarboxamido)-1H-b...)
Affinity DataIC50: 16nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274706(4-cyano-N-(5-(N-methylcyclohexanecarboxamido)-1-(3...)
Affinity DataIC50: 18nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM26813(N-[(2E)-5-[benzene(methyl)amido]-1-(2-carbamoyleth...)
Affinity DataIC50: 20nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274248(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 25nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274395(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 35nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274557(4-cyano-N-(1-isopropyl-5-(N-methylcyclohexanecarbo...)
Affinity DataIC50: 35nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274205(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 40nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274004(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclopropane...)
Affinity DataIC50: 46nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274394(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 56nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274752(N-(1-(3-amino-3-oxopropyl)-5-(N-methylacetamido)-1...)
Affinity DataIC50: 59nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274670(4-cyano-N-(5-(N-methylcyclohexanecarboxamido)-1-(2...)
Affinity DataIC50: 61nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274472(4-acetyl-N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyc...)
Affinity DataIC50: 68nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274630(N-(1-(2-amino-2-oxoethyl)-5-(N-methylcyclohexaneca...)
Affinity DataIC50: 73nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274007(N-(1-(3-amino-3-oxopropyl)-5-(methylamino)-1H-benz...)
Affinity DataIC50: 76nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274592(N-(1-(4-methoxyphenethyl)-5-(N-methylcyclohexaneca...)
Affinity DataIC50: 89nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274338(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 95nMAssay Description:Inhibition of IRKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274470(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 125nMAssay Description:Inhibition of IRKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274205(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 140nMAssay Description:Inhibition of IRKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274751(N-(1-(3-amino-3-oxopropyl)-5-(N-isopropylcyclohexa...)
Affinity DataIC50: 150nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274754(N-(1-(3-amino-3-oxopropyl)-5-(N-methylisobutyramid...)
Affinity DataIC50: 220nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274249(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 235nMAssay Description:Inhibition of IRKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274473(methyl 4-((1-(3-amino-3-oxopropyl)-5-(N-methylcycl...)
Affinity DataIC50: 250nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274511(4-cyano-N-(1-methyl-5-(N-methylcyclohexanecarboxam...)
Affinity DataIC50: 270nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274753(N-(1-(3-amino-3-oxopropyl)-5-(N-methylpropionamido...)
Affinity DataIC50: 320nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274340(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 320nMAssay Description:Inhibition of human ITK expressed in chicken DT40 cells assessed as B cell receptor-stimulated calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274669(N-(1-(3-(1H-imidazol-1-yl)propyl)-5-(N-methylcyclo...)
Affinity DataIC50: 510nMAssay Description:Inhibition of human ITK expressed in chicken DT40 cells assessed as B cell receptor-stimulated calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274509(N1-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexane...)
Affinity DataIC50: 520nMAssay Description:Inhibition of ITK by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274341(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 550nMAssay Description:Inhibition of IRKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274394(N-(1-(3-amino-3-oxopropyl)-5-(N-methylcyclohexanec...)
Affinity DataIC50: 550nMAssay Description:Inhibition of IRKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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