Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 2942
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26236BDBM26236(CHEMBL487569 | N-[6-(3,5-dimethoxyphenyl)-2-(3,5-d...)
Affinity DataKi:  0.190nM ΔG°:  -54.9kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26250BDBM26250(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[6-(pyrrolid...)
Affinity DataKi:  0.260nM ΔG°:  -54.2kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26256BDBM26256(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[6-(4-methox...)
Affinity DataKi:  0.440nM ΔG°:  -52.9kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26255BDBM26255(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[6-(3-methox...)
Affinity DataKi:  0.470nM ΔG°:  -52.7kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26251BDBM26251(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[6-(piperidi...)
Affinity DataKi:  0.560nM ΔG°:  -52.3kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26235BDBM26235(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(2-fluoro-3-...)
Affinity DataKi:  0.600nM ΔG°:  -52.1kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26249BDBM26249(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[6-(dimethyl...)
Affinity DataKi:  0.610nM ΔG°:  -52.1kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26253BDBM26253(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[6-(4-methyl...)
Affinity DataKi:  0.710nM ΔG°:  -51.7kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26254BDBM26254(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-{6-[(2-metho...)
Affinity DataKi:  0.720nM ΔG°:  -51.7kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26247BDBM26247(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[6-(morpholi...)
Affinity DataKi:  0.830nM ΔG°:  -51.3kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26234BDBM26234(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(3-methoxyph...)
Affinity DataKi:  0.920nM ΔG°:  -51.1kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26241BDBM26241(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(5-methoxypy...)
Affinity DataKi:  1.80nM ΔG°:  -49.4kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26257BDBM26257(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[6-(4-hydrox...)
Affinity DataKi:  1.90nM ΔG°:  -49.3kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26252BDBM26252(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[6-(1,4-oxaz...)
Affinity DataKi:  2.30nM ΔG°:  -48.8kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26237BDBM26237(CHEMBL458242 | N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)...)
Affinity DataKi:  2.30nM ΔG°:  -48.8kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26238BDBM26238(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(5-hydroxypy...)
Affinity DataKi:  2.90nM ΔG°:  -48.2kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26245BDBM26245(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[5-(morpholi...)
Affinity DataKi:  3nM ΔG°:  -48.2kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26239BDBM26239(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[5-(2-methox...)
Affinity DataKi:  3.10nM ΔG°:  -48.1kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26240BDBM26240(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(5-methoxypy...)
Affinity DataKi:  4nM ΔG°:  -47.5kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26250BDBM26250(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[6-(pyrrolid...)
Affinity DataKi:  7.20nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26242BDBM26242(methyl N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(5-me...)
Affinity DataKi:  7.40nM ΔG°:  -45.9kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26243BDBM26243(ethyl N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(5-met...)
Affinity DataKi:  7.80nM ΔG°:  -45.8kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26248BDBM26248(N-[6-(6-aminopyridin-2-yl)-2-(3,5-dimethyl-1H-pyra...)
Affinity DataKi:  7.90nM ΔG°:  -45.8kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26246BDBM26246(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[2-(morpholi...)
Affinity DataKi:  12nM ΔG°:  -44.8kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26236BDBM26236(CHEMBL487569 | N-[6-(3,5-dimethoxyphenyl)-2-(3,5-d...)
Affinity DataKi:  22nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26251BDBM26251(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[6-(piperidi...)
Affinity DataKi:  31nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26255BDBM26255(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[6-(3-methox...)
Affinity DataKi:  34nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26233BDBM26233(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(pyridin-4-y...)
Affinity DataKi:  40nM ΔG°:  -41.8kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26254BDBM26254(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-{6-[(2-metho...)
Affinity DataKi:  55nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26234BDBM26234(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(3-methoxyph...)
Affinity DataKi:  65nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26241BDBM26241(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(5-methoxypy...)
Affinity DataKi:  70nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26249BDBM26249(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[6-(dimethyl...)
Affinity DataKi:  81nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26256BDBM26256(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[6-(4-methox...)
Affinity DataKi:  85nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26244BDBM26244(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[4-(morpholi...)
Affinity DataKi:  87nM ΔG°:  -39.9kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26231BDBM26231(CHEMBL487765 | N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)...)
Affinity DataKi:  87nM ΔG°:  -39.9kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26235BDBM26235(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(2-fluoro-3-...)
Affinity DataKi:  110nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26239BDBM26239(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[5-(2-methox...)
Affinity DataKi:  110nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26232BDBM26232(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(pyridin-3-y...)
Affinity DataKi:  120nM ΔG°:  -39.1kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26253BDBM26253(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[6-(4-methyl...)
Affinity DataKi:  120nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26247BDBM26247(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[6-(morpholi...)
Affinity DataKi:  130nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26237BDBM26237(CHEMBL458242 | N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)...)
Affinity DataKi:  190nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26238BDBM26238(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(5-hydroxypy...)
Affinity DataKi:  195nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26245BDBM26245(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[5-(morpholi...)
Affinity DataKi:  220nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26252BDBM26252(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[6-(1,4-oxaz...)
Affinity DataKi:  280nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26231BDBM26231(CHEMBL487765 | N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)...)
Affinity DataKi:  290nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26248BDBM26248(N-[6-(6-aminopyridin-2-yl)-2-(3,5-dimethyl-1H-pyra...)
Affinity DataKi:  440nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26257BDBM26257(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[6-(4-hydrox...)
Affinity DataKi:  470nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26246BDBM26246(N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-[2-(morpholi...)
Affinity DataKi:  580nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26243BDBM26243(ethyl N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(5-met...)
Affinity DataKi:  620nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Bioscience

LigandChemical structure of BindingDB Monomer ID 26242BDBM26242(methyl N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(5-me...)
Affinity DataKi:  780nMAssay Description:The membranes prepared from HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2009
Entry Details Article
PubMed
Displayed 1 to 50 (of 54 total ) | Next | Last >>
Jump to: