Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50041718
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413787BDBM50413787(CHEMBL449380)
Affinity DataKi:  0.282nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21221BDBM21221(2-Cl-IB-MECA | CHEMBL431733 | C-IBzA-MU | 2-chloro...)
Affinity DataKi:  0.380nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413786BDBM50413786(CHEMBL483954)
Affinity DataKi:  0.398nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413798BDBM50413798(CHEMBL488149)
Affinity DataKi:  0.676nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413804BDBM50413804(CHEMBL486171)
Affinity DataKi:  0.891nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413790BDBM50413790(CHEMBL483969)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413791BDBM50413791(CHEMBL483975)
Affinity DataKi:  1.62nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413816BDBM50413816(CHEMBL516346)
Affinity DataKi:  2.19nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413797BDBM50413797(CHEMBL488148)
Affinity DataKi:  2.24nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413817BDBM50413817(CHEMBL473502)
Affinity DataKi:  2.51nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413789BDBM50413789(CHEMBL521312)
Affinity DataKi:  2.82nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413803BDBM50413803(CHEMBL487754)
Affinity DataKi:  2.82nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413806BDBM50413806(CHEMBL486374)
Affinity DataKi:  2.95nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413807BDBM50413807(CHEMBL516058)
Affinity DataKi:  3.63nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413802BDBM50413802(CHEMBL488777)
Affinity DataKi:  4.27nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413799BDBM50413799(CHEMBL487334)
Affinity DataKi:  5.62nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413794BDBM50413794(CHEMBL390877)
Affinity DataKi:  17.4nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413808BDBM50413808(CHEMBL474509)
Affinity DataKi:  18.2nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413818BDBM50413818(CHEMBL474310)
Affinity DataKi:  27.5nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413819BDBM50413819(CHEMBL474311)
Affinity DataKi:  29.5nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413805BDBM50413805(CHEMBL486373)
Affinity DataKi:  41.7nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413795BDBM50413795(CHEMBL488147)
Affinity DataKi:  85.1nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413812BDBM50413812(CHEMBL475320)
Affinity DataKi:  309nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413815BDBM50413815(CHEMBL457481)
Affinity DataKi:  347nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413813BDBM50413813(CHEMBL513368)
Affinity DataKi:  355nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413796BDBM50413796(CHEMBL520247)
Affinity DataKi:  417nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413814BDBM50413814(CHEMBL472886)
Affinity DataKi:  437nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413811BDBM50413811(CHEMBL474510)
Affinity DataKi:  513nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413823BDBM50413823(CHEMBL514483)
Affinity DataKi:  631nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413809BDBM50413809(CHEMBL462540)
Affinity DataKi:  871nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413810BDBM50413810(CHEMBL500736)
Affinity DataKi:  1.45E+3nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413788BDBM50413788(CHEMBL483802)
Affinity DataKi:  1.51E+3nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413793BDBM50413793(CHEMBL483813)
Affinity DataKi:  2.69E+3nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413792BDBM50413792(CHEMBL485165)
Affinity DataKi:  3.47E+3nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413822BDBM50413822(CHEMBL485164)
Affinity DataKi:  3.89E+3nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413800BDBM50413800(CHEMBL488576)
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413801BDBM50413801(CHEMBL529896)
Affinity DataKi:  4.47E+3nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413820BDBM50413820(CHEMBL474917)
Affinity DataKi:  7.59E+3nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sobhasaria Engineering College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413821BDBM50413821(CHEMBL443926)
Affinity DataKi:  4.90E+4nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed