Compile Data Set for Download or QSAR
Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50027529
LigandChemical structure of BindingDB Monomer ID 50256157BDBM50256157(N-((5-chloro-8-hydroxyquinolin-7-yl)(2-chloropheny...)
Affinity DataIC50: 350nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256061BDBM50256061(N-((5-chloro-8-hydroxyquinolin-7-yl)(4-nitrophenyl...)
Affinity DataIC50: 460nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256102BDBM50256102(N-((5-chloro-8-hydroxyquinolin-7-yl)(3-nitrophenyl...)
Affinity DataIC50: 490nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256700BDBM50256700(2-(N-methyl-N-phenylamino)-N-((5-chloro-8-hydroxyq...)
Affinity DataIC50: 560nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256062BDBM50256062(N-((5-chloro-8-hydroxyquinolin-7-yl)(3-fluoropheny...)
Affinity DataIC50: 620nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256160BDBM50256160(N-((5-bromo-8-hydroxyquinolin-7-yl)(3-nitrophenyl)...)
Affinity DataIC50: 620nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256005BDBM50256005(2-(benzyloxy)-N-((5-chloro-8-hydroxyquinolin-7-yl)...)
Affinity DataIC50: 700nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50255999BDBM50255999(N-((5-chloro-8-hydroxyquinolin-7-yl)(p-tolyl)methy...)
Affinity DataIC50: 760nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256312BDBM50256312(2-(p-tolyloxy)-N-((5-chloro-8-hydroxyquinolin-7-yl...)
Affinity DataIC50: 770nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50255970BDBM50255970(N-((5-chloro-8-hydroxyquinolin-7-yl)(phenyl)methyl...)
Affinity DataIC50: 780nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256660BDBM50256660(2-(N-methyl-N-phenylamino)-N-((5-chloro-8-hydroxyq...)
Affinity DataIC50: 780nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256214BDBM50256214(N-((5-bromo-8-hydroxyquinolin-7-yl)(2-chlorophenyl...)
Affinity DataIC50: 800nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256701BDBM50256701(2-(N-benzyl-N-methylamino)-N-((5-chloro-8-hydroxyq...)
Affinity DataIC50: 820nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256063BDBM50256063(2-(benzyloxy)-N-((5-chloro-8-hydroxyquinolin-7-yl)...)
Affinity DataIC50: 830nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256105BDBM50256105(N-((5-chloro-8-hydroxyquinolin-7-yl)(2-(trifluorom...)
Affinity DataIC50: 830nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256060BDBM50256060(N-((5-chloro-8-hydroxyquinolin-7-yl)(4-chloropheny...)
Affinity DataIC50: 830nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256313BDBM50256313(2-(4-methoxyphenoxy)-N-((5-chloro-8-hydroxyquinoli...)
Affinity DataIC50: 940nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256215BDBM50256215(N-((2-chlorophenyl)(8-hydroxy-5-nitroquinolin-7-yl...)
Affinity DataIC50: 940nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50255973BDBM50255973(N-((5-chloro-8-hydroxyquinolin-7-yl)(2-chloropheny...)
Affinity DataIC50: 990nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256059BDBM50256059(N-((5-chloro-8-hydroxyquinolin-7-yl)(4-methoxyphen...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256611BDBM50256611(2-(4-cyanophenylamino)-N-((5-chloro-8-hydroxyquino...)
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256499BDBM50256499(2-(4-chlorophenoxy)-N-((5-chloro-8-hydroxyquinolin...)
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256662BDBM50256662(2-(4-acetylphenylamino)-N-((5-chloro-8-hydroxyquin...)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256610BDBM50256610(2-(4-acetylphenylamino)-N-((5-chloro-8-hydroxyquin...)
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256698BDBM50256698(2-(4-chloro-3-methylphenylamino)-N-((5-chloro-8-hy...)
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256158BDBM50256158(N-((5-chloro-8-hydroxyquinolin-7-yl)(2-nitrophenyl...)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256103BDBM50256103(N-((5-chloro-8-hydroxyquinolin-7-yl)(2-fluoropheny...)
Affinity DataIC50: 1.22E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256740BDBM50256740(2-(N-methyl-N-phenylamino)-N-((5-chloro-8-hydroxyq...)
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256661BDBM50256661(2-(benzyl(methyl)amino)-N-((5-chloro-8-hydroxyquin...)
Affinity DataIC50: 1.28E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50255974BDBM50255974(2-(benzyl(methyl)amino)-N-((5-chloro-8-hydroxyquin...)
Affinity DataIC50: 1.31E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256216BDBM50256216(N-((8-hydroxy-5-methylquinolin-7-yl)(3-nitrophenyl...)
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256500BDBM50256500(2-(3-(dimethylamino)phenoxy)-N-((5-chloro-8-hydrox...)
Affinity DataIC50: 1.33E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50255969BDBM50255969(N-((8-hydroxy-5-nitroquinolin-7-yl)(phenyl)methyl)...)
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256738BDBM50256738(2-(4-chloro-3-methylphenylamino)-N-((5-chloro-8-hy...)
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256741BDBM50256741(2-(N-benzyl-N-methylamino)-N-((5-chloro-8-hydroxyq...)
Affinity DataIC50: 1.44E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50255971BDBM50255971(2-(4-chloro-3-methylphenylamino)-N-((5-chloro-8-hy...)
Affinity DataIC50: 1.48E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256613BDBM50256613(2-(4-chloro-3-methylphenylamino)-N-((5-chloro-8-hy...)
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256376BDBM50256376(N-((5-chloro-8-hydroxyquinolin-7-yl)(3-nitrophenyl...)
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256314BDBM50256314(2-(3-(dimethylamino)phenoxy)-N-((5-chloro-8-hydrox...)
Affinity DataIC50: 1.67E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256739BDBM50256739(2-(benzylamino)-N-((5-chloro-8-hydroxyquinolin-7-y...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256556BDBM50256556(2-(3-(dimethylamino)phenoxy)-N-((5-chloro-8-hydrox...)
Affinity DataIC50: 1.72E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256659BDBM50256659(2-(benzylamino)-N-((5-chloro-8-hydroxyquinolin-7-y...)
Affinity DataIC50: 1.83E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256104BDBM50256104(N-((5-chloro-8-hydroxyquinolin-7-yl)(o-tolyl)methy...)
Affinity DataIC50: 1.85E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50255972BDBM50255972(2-(benzylamino)-N-((5-chloro-8-hydroxyquinolin-7-y...)
Affinity DataIC50: 1.89E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256102BDBM50256102(N-((5-chloro-8-hydroxyquinolin-7-yl)(3-nitrophenyl...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of ADAMTS4 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256429BDBM50256429(2-(p-tolyloxy)-N-((5-chloro-8-hydroxyquinolin-7-yl...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256612BDBM50256612(2-(3-(dimethylamino)phenylamino)-N-((5-chloro-8-hy...)
Affinity DataIC50: 1.93E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50255967BDBM50255967(N-((8-hydroxyquinolin-7-yl)(phenyl)methyl)-2-pheno...)
Affinity DataIC50: 2.28E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256159BDBM50256159(N-((5-chloro-8-hydroxyquinolin-7-yl)(2-cyanophenyl...)
Affinity DataIC50: 2.32E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256426BDBM50256426(2-(4-Acetyl-phenoxy)-N-[(5-chloro-8-hydroxy-quinol...)
Affinity DataIC50: 2.33E+3nMAssay Description:Inhibition of ADAMTS5 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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