Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50027549
TargetE3 ubiquitin-protein ligase Mdm2(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273917BDBM50273917(Isolissoclinotoxin B | CHEMBL462089)
Affinity DataIC50: 5.86E+4nMAssay Description:Inhibition of GST fused human Hdm2 assessed as polyubiquitylation by electrochemiluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273972BDBM50273972(Lissoclinidine B | CHEMBL461462)
Affinity DataIC50: 5.86E+4nMAssay Description:Inhibition of GST fused human Hdm2 assessed as polyubiquitylation by electrochemiluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273919BDBM50273919(Diplamine B | CHEMBL513108)
Affinity DataIC50: 1.01E+5nMAssay Description:Inhibition of GST fused human Hdm2 assessed as polyubiquitylation by electrochemiluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50273918BDBM50273918(N,N-dimethyl-5-methylvaracin | CHEMBL462090)
Affinity DataIC50: 1.21E+5nMAssay Description:Inhibition of GST fused human Hdm2 assessed as polyubiquitylation by electrochemiluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50240848BDBM50240848(2-(3,4-Dimethoxy-5,6,7,8,9-pentathia-benzocyclohep...)
Affinity DataIC50: 2.95E+5nMAssay Description:Inhibition of GST fused human Hdm2 assessed as polyubiquitylation by electrochemiluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed