Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50027670
TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50254947(MPrP | CHEMBL481189)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human ERalpha receptor expressed in HEC1 cells assessed as transcriptional activation after 24 hrs by luciferase reporter gene...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50254908(4-[1-(4-hydroxyphenyl)-4-methyl-5-{4-[2-(piperidin...)
Affinity DataIC50: 80nMAssay Description:Antagonist activity at human ERalpha receptor expressed in HEC1 cells assessed as transcriptional activation after 24 hrs by luciferase reporter gene...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50254948((2E)-3-{4-[1,3-bis(4-hydroxyphenyl)-4-methyl-1H-py...)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human ERalpha receptor expressed in HEC1 cells assessed as transcriptional activation after 24 hrs by luciferase reporter gene...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed