Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50027680
LigandPNGBDBM50255048(3,4-Difluoro-2-(2-fluoro-4-iodo-phenylamino)-5-[(5...)
Affinity DataIC50: 100nMAssay Description:Binding affinity to SRCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255048(3,4-Difluoro-2-(2-fluoro-4-iodo-phenylamino)-5-[(5...)
Affinity DataIC50: 300nMAssay Description:Binding affinity to ABLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255048(3,4-Difluoro-2-(2-fluoro-4-iodo-phenylamino)-5-[(5...)
Affinity DataIC50: 500nMAssay Description:Binding affinity to LCKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255012(5-((4-(methylsulfonyl)benzylamino)methyl)-3,4-difl...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity to Aurora AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50255012(5-((4-(methylsulfonyl)benzylamino)methyl)-3,4-difl...)
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity to TRAK-AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255013((S)-5-((2,4-diamino-4-oxobutanamido)methyl)-3,4-di...)
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity to PKC beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255048(3,4-Difluoro-2-(2-fluoro-4-iodo-phenylamino)-5-[(5...)
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity to FGFR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255013((S)-5-((2,4-diamino-4-oxobutanamido)methyl)-3,4-di...)
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity to Aurora AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50255048(3,4-Difluoro-2-(2-fluoro-4-iodo-phenylamino)-5-[(5...)
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity to VEGFR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50255049(5-{[2-(4-Chloro-benzenesulfonyl)-acetyl]-hydrazono...)
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity to SRCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEphrin type-A receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255048(3,4-Difluoro-2-(2-fluoro-4-iodo-phenylamino)-5-[(5...)
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity to ECKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255049(5-{[2-(4-Chloro-benzenesulfonyl)-acetyl]-hydrazono...)
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity to CLK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255048(3,4-Difluoro-2-(2-fluoro-4-iodo-phenylamino)-5-[(5...)
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity to Aurora AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50255048(3,4-Difluoro-2-(2-fluoro-4-iodo-phenylamino)-5-[(5...)
Affinity DataIC50: 4.00E+3nMAssay Description:Binding affinity to MAP3K9More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50255013((S)-5-((2,4-diamino-4-oxobutanamido)methyl)-3,4-di...)
Affinity DataIC50: 4.00E+3nMAssay Description:Binding affinity to SRCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255049(5-{[2-(4-Chloro-benzenesulfonyl)-acetyl]-hydrazono...)
Affinity DataIC50: 4.00E+3nMAssay Description:Binding affinity to ABLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255049(5-{[2-(4-Chloro-benzenesulfonyl)-acetyl]-hydrazono...)
Affinity DataIC50: 4.00E+3nMAssay Description:Binding affinity to Aurora AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50255049(5-{[2-(4-Chloro-benzenesulfonyl)-acetyl]-hydrazono...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity to TRAK-AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50255012(5-((4-(methylsulfonyl)benzylamino)methyl)-3,4-difl...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity to MAP3K9More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255013((S)-5-((2,4-diamino-4-oxobutanamido)methyl)-3,4-di...)
Affinity DataIC50: 6.00E+3nMAssay Description:Binding affinity to MST2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255049(5-{[2-(4-Chloro-benzenesulfonyl)-acetyl]-hydrazono...)
Affinity DataIC50: 7.00E+3nMAssay Description:Binding affinity to LCKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50255049(5-{[2-(4-Chloro-benzenesulfonyl)-acetyl]-hydrazono...)
Affinity DataIC50: 7.00E+3nMAssay Description:Binding affinity to MAP3K9More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255048(3,4-Difluoro-2-(2-fluoro-4-iodo-phenylamino)-5-[(5...)
Affinity DataIC50: 7.00E+3nMAssay Description:Binding affinity to BTKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50255013((S)-5-((2,4-diamino-4-oxobutanamido)methyl)-3,4-di...)
Affinity DataIC50: 1.30E+4nMAssay Description:Binding affinity to TRAK-AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255048(3,4-Difluoro-2-(2-fluoro-4-iodo-phenylamino)-5-[(5...)
Affinity DataIC50: 1.50E+4nMAssay Description:Binding affinity to CLK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50255012(5-((4-(methylsulfonyl)benzylamino)methyl)-3,4-difl...)
Affinity DataIC50: 1.80E+4nMAssay Description:Binding affinity to VEGFR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50255048(3,4-Difluoro-2-(2-fluoro-4-iodo-phenylamino)-5-[(5...)
Affinity DataIC50: 2.00E+4nMAssay Description:Binding affinity to TRAK-AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255012(5-((4-(methylsulfonyl)benzylamino)methyl)-3,4-difl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to PKC beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255049(5-{[2-(4-Chloro-benzenesulfonyl)-acetyl]-hydrazono...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to PKC beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255048(3,4-Difluoro-2-(2-fluoro-4-iodo-phenylamino)-5-[(5...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to PKC beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255012(5-((4-(methylsulfonyl)benzylamino)methyl)-3,4-difl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to MST2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255049(5-{[2-(4-Chloro-benzenesulfonyl)-acetyl]-hydrazono...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to MST2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255048(3,4-Difluoro-2-(2-fluoro-4-iodo-phenylamino)-5-[(5...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to MST2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50255012(5-((4-(methylsulfonyl)benzylamino)methyl)-3,4-difl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to SRCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255013((S)-5-((2,4-diamino-4-oxobutanamido)methyl)-3,4-di...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to ABLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255012(5-((4-(methylsulfonyl)benzylamino)methyl)-3,4-difl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to ABLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255013((S)-5-((2,4-diamino-4-oxobutanamido)methyl)-3,4-di...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to LCKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255012(5-((4-(methylsulfonyl)benzylamino)methyl)-3,4-difl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to LCKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255013((S)-5-((2,4-diamino-4-oxobutanamido)methyl)-3,4-di...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to FGFR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255012(5-((4-(methylsulfonyl)benzylamino)methyl)-3,4-difl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to FGFR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255049(5-{[2-(4-Chloro-benzenesulfonyl)-acetyl]-hydrazono...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to FGFR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEphrin type-A receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255013((S)-5-((2,4-diamino-4-oxobutanamido)methyl)-3,4-di...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to ECKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEphrin type-A receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255012(5-((4-(methylsulfonyl)benzylamino)methyl)-3,4-difl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to ECKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetEphrin type-A receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255049(5-{[2-(4-Chloro-benzenesulfonyl)-acetyl]-hydrazono...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to ECKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50255013((S)-5-((2,4-diamino-4-oxobutanamido)methyl)-3,4-di...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to VEGFR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50255049(5-{[2-(4-Chloro-benzenesulfonyl)-acetyl]-hydrazono...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to VEGFR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50255013((S)-5-((2,4-diamino-4-oxobutanamido)methyl)-3,4-di...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to MAP3K9More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255013((S)-5-((2,4-diamino-4-oxobutanamido)methyl)-3,4-di...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to BTKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255012(5-((4-(methylsulfonyl)benzylamino)methyl)-3,4-difl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to BTKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50255049(5-{[2-(4-Chloro-benzenesulfonyl)-acetyl]-hydrazono...)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to BTKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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