Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50041721
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50135878BDBM50135878((R)-1-phenyl-2-(o-tolyloxy)ethanamine | (R)-1-Phen...)
Affinity DataEC50:  1.00E+3nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413853BDBM50413853(CHEMBL485004)
Affinity DataEC50:  1.70E+3nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413870BDBM50413870(CHEMBL444700)
Affinity DataEC50:  1.91E+3nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413854BDBM50413854(CHEMBL486721)
Affinity DataEC50:  2.29E+3nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413858BDBM50413858(CHEMBL487338)
Affinity DataEC50:  2.40E+3nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413869BDBM50413869(CHEMBL448542)
Affinity DataEC50:  2.69E+3nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413860BDBM50413860(CHEMBL501561)
Affinity DataEC50:  2.88E+3nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413862BDBM50413862(CHEMBL486528)
Affinity DataEC50:  3.02E+3nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50135873BDBM50135873((S)-2-(4-chlorophenoxy)-1-phenylethanamine | (S)-2...)
Affinity DataEC50:  3.02E+3nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50135880BDBM50135880((S)-2-(2,6-Dimethyl-phenoxy)-1-phenyl-ethylamine |...)
Affinity DataEC50:  3.02E+3nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50135886BDBM50135886((R)-2-(2,6-Dimethyl-phenoxy)-1-phenyl-ethylamine |...)
Affinity DataEC50:  3.02E+3nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413859BDBM50413859(CHEMBL486315)
Affinity DataEC50:  3.72E+3nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50135874BDBM50135874((R)-2-phenoxy-1-phenylethanamine | (R)-2-Phenoxy-1...)
Affinity DataEC50:  3.98E+3nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413868BDBM50413868(CHEMBL452986)
Affinity DataEC50:  4.68E+3nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413856BDBM50413856(CHEMBL446777)
Affinity DataEC50:  5.75E+3nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413857BDBM50413857(CHEMBL474672)
Affinity DataEC50:  5.75E+3nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413867BDBM50413867(CHEMBL483784)
Affinity DataEC50:  7.08E+3nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50135882BDBM50135882((S)-2-(4-chloro-2,6-dimethylphenoxy)-1-phenylethan...)
Affinity DataEC50:  7.94E+3nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413842BDBM50413842(CHEMBL473498)
Affinity DataEC50:  9.12E+3nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50135881BDBM50135881((R)-2-(4-chlorophenoxy)-1-phenylethanamine | (R)-2...)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413852BDBM50413852(CHEMBL485003)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413841BDBM50413841(CHEMBL472884)
Affinity DataEC50:  1.12E+4nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413843BDBM50413843(CHEMBL502686)
Affinity DataEC50:  1.20E+4nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50135885BDBM50135885((R)-2-(4-Chloro-2-methyl-phenoxy)-1-phenyl-ethylam...)
Affinity DataEC50:  1.51E+4nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50135879BDBM50135879((S)-2-phenoxy-1-phenylethanamine | (S)-2-Phenoxy-1...)
Affinity DataEC50:  1.58E+4nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413866BDBM50413866(CHEMBL485647)
Affinity DataEC50:  1.74E+4nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50135877BDBM50135877((R)-2-(4-Chloro-2,6-dimethyl-phenoxy)-1-phenyl-eth...)
Affinity DataEC50:  1.95E+4nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50135883BDBM50135883((R)-1-(2,6-dimethylphenoxy)propan-2-amine | (2R)-1...)
Affinity DataEC50:  2.29E+4nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413861BDBM50413861(CHEMBL486414)
Affinity DataEC50:  2.29E+4nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413865BDBM50413865(CHEMBL468775)
Affinity DataEC50:  2.34E+4nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50135884BDBM50135884((S)-1-(2,6-dimethylphenoxy)propan-2-amine | (S)-2-...)
Affinity DataEC50:  2.69E+4nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413846BDBM50413846(CHEMBL473706)
Affinity DataEC50:  2.82E+4nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413851BDBM50413851(CHEMBL519199)
Affinity DataEC50:  3.16E+4nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413844BDBM50413844(CHEMBL473499)
Affinity DataEC50:  4.07E+4nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413848BDBM50413848(CHEMBL484996)
Affinity DataEC50:  6.76E+4nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413845BDBM50413845(CHEMBL473705)
Affinity DataEC50:  6.76E+4nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413850BDBM50413850(CHEMBL485002)
Affinity DataEC50:  2.00E+5nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413863BDBM50413863(CHEMBL2021482)
Affinity DataEC50:  2.09E+5nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413847BDBM50413847(CHEMBL484981)
Affinity DataEC50:  2.19E+5nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50291989BDBM50291989(CHEMBL387108 | (S)-2-amino-N-(2,6-dimethylphenyl)p...)
Affinity DataEC50:  2.24E+5nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413864BDBM50413864(CHEMBL2021481)
Affinity DataEC50:  2.34E+5nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50291990BDBM50291990(CHEMBL222944 | Tonocard | 2-Amino-N-(2,6-dimethyl-...)
Affinity DataEC50:  2.75E+5nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413855BDBM50413855(CHEMBL501346)
Affinity DataEC50:  5.01E+5nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50413849BDBM50413849(CHEMBL484833)
Affinity DataEC50:  5.01E+5nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed