Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 3086
LigandChemical structure of BindingDB Monomer ID 27826BDBM27826(4-fluoro-2-[(2-{[2-methoxy-4-(1-propylpiperidin-4-...)
Affinity DataIC50: 0.300nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27825BDBM27825(4-fluoro-2-[(2-{[2-methoxy-4-(1-propylpiperidin-3-...)
Affinity DataIC50: 0.400nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27842BDBM27842(4,5-difluoro-2-{[2-({2-methoxy-4-[4-(propan-2-yl)p...)
Affinity DataIC50: 0.5nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27822BDBM27822(2-[(2-{[2-methoxy-4-(1-propyl-1,2,5,6-tetrahydropy...)
Affinity DataIC50: 0.600nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27839BDBM27839(CHEMBL458865 | 5-fluoro-2-{[2-({2-methoxy-4-[4-(pr...)
Affinity DataIC50: 0.800nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27828BDBM27828(4-fluoro-2-{[2-({2-methoxy-4-[4-(propan-2-yl)piper...)
Affinity DataIC50: 0.800nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27841BDBM27841(2,4-difluoro-6-{[2-({2-methoxy-4-[4-(propan-2-yl)p...)
Affinity DataIC50: 0.800nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27823BDBM27823(4-fluoro-2-[(2-{[2-methoxy-4-(1-propyl-1,2,5,6-tet...)
Affinity DataIC50: 0.800nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27838BDBM27838(2-{[2-({2-methoxy-4-[4-(propan-2-yl)piperazin-1-yl...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27840BDBM27840(CHEMBL463932 | 2,3-difluoro-6-{[2-({2-methoxy-4-[4...)
Affinity DataIC50: 1.30nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27827BDBM27827(4-fluoro-2-[(2-{[2-methoxy-4-(4-propylpiperazin-1-...)
Affinity DataIC50: 1.60nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27829BDBM27829(4-fluoro-2-[(2-{[2-methoxy-4-(morpholin-4-yl)pheny...)
Affinity DataIC50: 1.60nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27819BDBM27819(2-[(2-{[4-(1-propyl-1,2,5,6-tetrahydropyridin-3-yl...)
Affinity DataIC50: 1.60nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27820BDBM27820(2-[(2-{[2-fluoro-4-(1-propyl-1,2,5,6-tetrahydropyr...)
Affinity DataIC50: 1.60nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27835BDBM27835(2-{[2-({5-chloro-2-methoxy-4-[4-(propan-2-yl)piper...)
Affinity DataIC50: 1.60nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27783BDBM27783(CHEMBL507625 | BMCL19469 Compound 13 | 2-fluoro-6-...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27833BDBM27833(2-fluoro-6-{[2-({5-fluoro-2-methoxy-4-[4-(propan-2...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27834BDBM27834(2-fluoro-6-{[2-({2-methoxy-5-methyl-4-[4-(propan-2...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27844BDBM27844(5-fluoro-2-{[2-({2-methoxy-4-[4-(propan-2-yl)piper...)
Affinity DataIC50: 3.20nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27832BDBM27832(2-{[2-({2,5-dimethoxy-4-[4-(propan-2-yl)piperazin-...)
Affinity DataIC50: 3.20nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27824BDBM27824(4-fluoro-2-[(2-{[2-(propan-2-yloxy)-4-(1-propyl-1,...)
Affinity DataIC50: 3.20nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27836BDBM27836(2-fluoro-6-{[2-({3-fluoro-2-methoxy-4-[4-(propan-2...)
Affinity DataIC50: 4nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27784BDBM27784(2-fluoro-6-{[2-({2-methoxy-5-[4-(propan-2-yl)piper...)
Affinity DataIC50: 4nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27843BDBM27843(2-fluoro-6-{[2-({2-methoxy-4-[4-(propan-2-yl)piper...)
Affinity DataIC50: 5nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27818BDBM27818(2-[(2-{[2-methyl-4-(1-propyl-1,2,5,6-tetrahydropyr...)
Affinity DataIC50: 5nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27847BDBM27847(5-fluoro-N-(2-hydroxyethyl)-2-{[2-({2-methoxy-4-[4...)
Affinity DataIC50: 5nMAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27845BDBM27845(5-fluoro-N-hydroxy-2-{[2-({2-methoxy-4-[4-(propan-...)
Affinity DataIC50: 6.30nMAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27837BDBM27837(2-fluoro-6-{[2-({2-methoxy-3-methyl-4-[4-(propan-2...)
Affinity DataIC50: 8nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27846BDBM27846(N-[(2R)-2,3-dihydroxypropyl]-5-fluoro-2-{[2-({2-me...)
Affinity DataIC50: 16nMAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27821BDBM27821(2-[(2-{[4-(1-propyl-1,2,5,6-tetrahydropyridin-3-yl...)
Affinity DataIC50: 20nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27785BDBM27785(2-fluoro-6-{[2-({2-methoxy-4-methyl-5-[4-(propan-2...)
Affinity DataIC50: 20nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27848BDBM27848(5-fluoro-2-{[2-({2-methoxy-4-[4-(propan-2-yl)piper...)
Affinity DataIC50: 25nMAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27830BDBM27830(2-fluoro-6-{[2-({2-methoxy-4-[4-(propan-2-yl)piper...)
Affinity DataIC50: 50nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 27831BDBM27831(2-fluoro-6-{[2-({2-methoxy-4-[4-(propan-2-yl)piper...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Assays are performed in 384-well microtiter plates in reaction buffer containing biotinylated substrate, ATP, and purified activated GST-IGF-1R in th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2009
Entry Details Article
PubMed