Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50027858
TargetTranscription factor Jun(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development Centre

Curated by ChEMBL
LigandPNGBDBM50279429(3-(4-Chloro-phenyl)-2-(4-methyl-2-methylamino-thia...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of AP1 (unknown origin) expressed in HEK293 cells assessed as inhibition of TNFalpha-induced transcriptional activation treated 24 hrs bef...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development Centre

Curated by ChEMBL
LigandPNGBDBM50279431(3-(4-Chloro-phenyl)-2-[2-(4-chloro-phenylamino)-4-...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of AP1 (unknown origin) expressed in HEK293 cells assessed as inhibition of TNFalpha-induced transcriptional activation treated 24 hrs bef...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development Centre

Curated by ChEMBL
LigandPNGBDBM50279698(2-(4-Methyl-2-methylamino-thiazol-5-yl)-3-o-tolyl-...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of AP1 (unknown origin) expressed in HEK293 cells assessed as inhibition of TNFalpha-induced transcriptional activation treated 24 hrs bef...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
B.V. Patel Pharmaceutical Education And Research Development Centre

Curated by ChEMBL
LigandPNGBDBM50279699(2-(4-Methyl-2-phenylamino-thiazol-5-yl)-3-o-tolyl-...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of AP1 (unknown origin) expressed in HEK293 cells assessed as inhibition of TNFalpha-induced transcriptional activation treated 24 hrs bef...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed