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Found 22 Enz. Inhib. hit(s) with all data for entry = 50038891
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295565(3-[4'-(4''-Bromophenyl)benzoyl]-3,4-dihydro-8-meth...)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibition of mouse iNOS expressed in insect Sf9 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295567(3-[4'-(4''-Methoxyphenyl)benzoyl]-3,4-dihydro-8-me...)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibition of mouse iNOS expressed in insect Sf9 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295568(3,4-Dihydro-8-methyl-3-[2-(6-methylnaphthoyl)]-2H-...)
Affinity DataKi:  2.30E+4nMAssay Description:Inhibition of mouse iNOS expressed in insect Sf9 cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295566(3-[4'-(4''-Cyanophenyl)benzoyl]-3,4-dihydro-8-meth...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of mouse recombinant iNOS expressed in Escherichia coli assessed as NADPH consumption after 2 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295566(3-[4'-(4''-Cyanophenyl)benzoyl]-3,4-dihydro-8-meth...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of bovine recombinant eNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioacti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295571(3-[4'-(4''-Chlorobenzyloxy)benzoyl]-3,4-dihydro-8-...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of bovine recombinant eNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioacti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295567(3-[4'-(4''-Methoxyphenyl)benzoyl]-3,4-dihydro-8-me...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of mouse recombinant iNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioactiv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50209245(CHEMBL247378)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of rat recombinant nNOS expressed in Saccharomyces cerevisiae assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295565(3-[4'-(4''-Bromophenyl)benzoyl]-3,4-dihydro-8-meth...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of mouse recombinant iNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioactiv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295568(3,4-Dihydro-8-methyl-3-[2-(6-methylnaphthoyl)]-2H-...)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of mouse recombinant iNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioactiv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295565(3-[4'-(4''-Bromophenyl)benzoyl]-3,4-dihydro-8-meth...)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of mouse recombinant iNOS expressed in Escherichia coli assessed as NADPH consumption after 2 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295570(3,4-Dihydro-6,8-dimethyl-3-[2-(6-methylnaphthoyl)]...)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of mouse recombinant iNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioactiv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50209245(CHEMBL247378)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of mouse recombinant iNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioactiv...More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50209245(CHEMBL247378)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibition of bovine recombinant eNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioacti...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295566(3-[4'-(4''-Cyanophenyl)benzoyl]-3,4-dihydro-8-meth...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of mouse recombinant iNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioactiv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295570(3,4-Dihydro-6,8-dimethyl-3-[2-(6-methylnaphthoyl)]...)
Affinity DataIC50:  5.30E+4nMAssay Description:Inhibition of bovine recombinant eNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioacti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295567(3-[4'-(4''-Methoxyphenyl)benzoyl]-3,4-dihydro-8-me...)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of bovine recombinant eNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioacti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295570(3,4-Dihydro-6,8-dimethyl-3-[2-(6-methylnaphthoyl)]...)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of rat recombinant nNOS expressed in Saccharomyces cerevisiae assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295567(3-[4'-(4''-Methoxyphenyl)benzoyl]-3,4-dihydro-8-me...)
Affinity DataIC50:  8.70E+4nMAssay Description:Inhibition of rat recombinant nNOS expressed in Saccharomyces cerevisiae assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295569(3-[4'-(4''-Bromophenyl)benzoyl]-3,4-dihydro-6,8-di...)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibition of mouse recombinant iNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioactiv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295566(3-[4'-(4''-Cyanophenyl)benzoyl]-3,4-dihydro-8-meth...)
Affinity DataIC50:  1.28E+5nMAssay Description:Inhibition of rat recombinant nNOS expressed in Saccharomyces cerevisiae assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Bos taurus (bovine))
Christian-Albrechts-University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50295569(3-[4'-(4''-Bromophenyl)benzoyl]-3,4-dihydro-6,8-di...)
Affinity DataIC50:  1.88E+5nMAssay Description:Inhibition of bovine recombinant eNOS expressed in Escherichia coli assessed as conversion of [gamma-14C]L-arginine to [14C]L-citrulline by radioacti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed