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Found 11 Enz. Inhib. hit(s) with all data for entry = 50028164
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Institute Of Biochemistry And Biophysics

Curated by ChEMBL
LigandPNGBDBM50276678(3-(4,5,6,7-Tetrabromo-1H-1,2,3-benzotriazol-1-yl)p...)
Affinity DataIC50:  320nMAssay Description:Inhibition of human recombinant casein kinase 2 subunit alpha expressed in Escherichia coli BL21 (DE3) assessed as [32P] incorporation by liquid scin...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Institute Of Biochemistry And Biophysics

Curated by ChEMBL
LigandPNGBDBM50276679(3-(4,5,6,7-Tetrabromo-2H-1,2,3-benzotriazol-2-yl)p...)
Affinity DataIC50:  340nMAssay Description:Inhibition of human recombinant casein kinase 2 subunit alpha expressed in Escherichia coli BL21 (DE3) assessed as [32P] incorporation by liquid scin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Institute Of Biochemistry And Biophysics

Curated by ChEMBL
LigandPNGBDBM11323(4,5,6,7-tetrabromo-1H-1,2,3-benzotriazole | 4,5,6,...)
Affinity DataIC50:  500nMAssay Description:Inhibition of human recombinant casein kinase 2 subunit alpha expressed in Escherichia coli BL21 (DE3) assessed as [32P] incorporation by liquid scin...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Institute Of Biochemistry And Biophysics

Curated by ChEMBL
LigandPNGBDBM50276732(3-(4,5,6,7-Tetrabromo-1H-benzimidazol-1-yl)propan-...)
Affinity DataIC50:  540nMAssay Description:Inhibition of human recombinant casein kinase 2 subunit alpha expressed in Escherichia coli BL21 (DE3) assessed as [32P] incorporation by liquid scin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Institute Of Biochemistry And Biophysics

Curated by ChEMBL
LigandPNGBDBM50156669(4,5,6,7-TETRABROMO-BENZIMIDAZOLE | 4,5,6,7-tetrabr...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human recombinant casein kinase 2 subunit alpha expressed in Escherichia coli BL21 (DE3) assessed as [32P] incorporation by liquid scin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Institute Of Biochemistry And Biophysics

Curated by ChEMBL
LigandPNGBDBM50276731(4-(4,5,6,7-tetrabromo-2H-1,2,3-benzotriazol-2-yl)b...)
Affinity DataIC50:  1.73E+3nMAssay Description:Inhibition of human recombinant casein kinase 2 subunit alpha expressed in Escherichia coli BL21 (DE3) assessed as [32P] incorporation by liquid scin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Institute Of Biochemistry And Biophysics

Curated by ChEMBL
LigandPNGBDBM50276680(3-(4,5,6,7-Tetrabromo-2H-1,2,3-benzotriazol-2-yl)p...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human recombinant casein kinase 2 subunit alpha expressed in Escherichia coli BL21 (DE3) assessed as [32P] incorporation by liquid scin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Institute Of Biochemistry And Biophysics

Curated by ChEMBL
LigandPNGBDBM50276733(1-(3-chloropropyl)-4,5,6,7-tetrabromo-1H-benzimida...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of human recombinant casein kinase 2 subunit alpha expressed in Escherichia coli BL21 (DE3) assessed as [32P] incorporation by liquid scin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Institute Of Biochemistry And Biophysics

Curated by ChEMBL
LigandPNGBDBM50276730(4,5,6,7-Tetrabromo-2-[3-(4-methylpiperazin-1-yl)pr...)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of human recombinant casein kinase 2 subunit alpha expressed in Escherichia coli BL21 (DE3) assessed as [32P] incorporation by liquid scin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Institute Of Biochemistry And Biophysics

Curated by ChEMBL
LigandPNGBDBM50276630(2-(perbromo-1H-benzo[d][1,2,3]triazol-1-yl)ethanol...)
Affinity DataIC50:  9.25E+3nMAssay Description:Inhibition of human recombinant casein kinase 2 subunit alpha expressed in Escherichia coli BL21 (DE3) assessed as [32P] incorporation by liquid scin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Institute Of Biochemistry And Biophysics

Curated by ChEMBL
LigandPNGBDBM50276682(4,5,6,7-Tetrabromo-1-[3-(4-methylpiperazin-1-yl)pr...)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibition of human recombinant casein kinase 2 subunit alpha expressed in Escherichia coli BL21 (DE3) assessed as [32P] incorporation by liquid scin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed