Affinity DataIC50: 19.9nMAssay Description:Antagonist activity at human recombinant C5a receptor in HEK cells assessed as inhibition of C5a-induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataIC50: 25.1nMAssay Description:Antagonist activity at human recombinant C5a receptor in HEK cells assessed as inhibition of C5a-induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataIC50: 31.6nMAssay Description:Displacement of [Alexa647]C5a from human recombinant C5a receptor expressed in HEK cells by membrane binding assay in presence of [35S]GTPgammaSMore data for this Ligand-Target Pair
Affinity DataIC50: 39.8nMAssay Description:Antagonist activity at human recombinant C5a receptor in HEK cells assessed as inhibition of C5a-induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataIC50: 39.8nMAssay Description:Displacement of [Alexa647]C5a from human recombinant C5a receptor expressed in HEK cells by whole cell binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 63.1nMAssay Description:Antagonist activity at human recombinant C5a receptor in HEK cells assessed as inhibition of C5a-induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataIC50: 79.4nMAssay Description:Displacement of [Alexa647]C5a from human recombinant C5a receptor expressed in HEK cells by whole cell binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human recombinant C5a receptor in HEK cells assessed as inhibition of C5a-induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataIC50: >100nMAssay Description:Antagonist activity at human recombinant C5a receptor in HEK cells assessed as inhibition of C5a-induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Antagonist activity at human recombinant C5a receptor in HEK cells assessed as inhibition of C5a-induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Antagonist activity at human recombinant C5a receptor in HEK cells assessed as inhibition of C5a-induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Displacement of [Alexa647]C5a from human recombinant C5a receptor expressed in HEK cells by membrane binding assay in presence of [35S]GTPgammaSMore data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Antagonist activity at human recombinant C5a receptor in HEK cells assessed as inhibition of C5a-induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataIC50: 794nMAssay Description:Displacement of [Alexa647]C5a from human recombinant C5a receptor expressed in HEK cells by membrane binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 794nMAssay Description:Antagonist activity at human recombinant C5a receptor in HEK cells assessed as inhibition of C5a-induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human recombinant C5a receptor in HEK cells assessed as inhibition of C5a-induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataIC50: 3.16E+3nMAssay Description:Displacement of [Alexa647]C5a from human recombinant C5a receptor expressed in HEK cells by membrane binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.16E+3nMAssay Description:Antagonist activity at human recombinant C5a receptor in HEK cells assessed as inhibition of C5a-induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human recombinant C5a receptor in HEK cells assessed as inhibition of C5a-induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human recombinant C5a receptor in HEK cells assessed as inhibition of C5a-induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human recombinant C5a receptor in HEK cells assessed as inhibition of C5a-induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 123nMAssay Description:Antagonist activity at human recombinant C5a receptor expressed in HEK cells assessed as inhibition of C5a-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair