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Found
89
Enz. Inhib. hit(s) with all data for entry = 50031610
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316184
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((S)-3-amino...)
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Affinity Data
Ki: 0.200nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316183
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((R)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.200nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316192
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((R)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.400nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316183
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((R)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.600nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM25013
(4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3S...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316192
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((R)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-beta serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316184
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((S)-3-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1nM
Assay Description:
Inhibition of AKT2
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-gamma serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316192
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((R)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1nM
Assay Description:
Inhibition of AKT3
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316185
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((R)-3-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.90nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-beta serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316183
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((R)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 2nM
Assay Description:
Inhibition of AKT2
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316184
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((S)-3-amino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM25013
(4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3S...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316195
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((dimethylam...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316194
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-6-((me...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 3nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316187
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-(3-aminoprop...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 3nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316182
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 3nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316201
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 3nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-gamma serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316183
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((R)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 3nM
Assay Description:
Inhibition of AKT3
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316182
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 3nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316190
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((R)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 3nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316185
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((R)-3-amino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-beta serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM25013
(4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3S...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 4nM
Assay Description:
Inhibition of AKT2
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316193
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-(2-aminoethy...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-beta serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316192
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((R)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 5nM
Assay Description:
Inhibition of AKT2
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316189
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-(2-aminoetho...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316191
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316189
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-(2-aminoetho...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 6nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316186
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-(aminomethyl...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316188
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-6-(pyr...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316199
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((R)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 8nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-gamma serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM25013
(4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3S...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 9nM
Assay Description:
Inhibition of AKT3
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-beta serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316183
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((R)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 10nM
Assay Description:
Inhibition of AKT2
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316198
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-6-(2-(...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 12nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-beta serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM25013
(4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3S...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 13nM
Assay Description:
Inhibition of AKT2
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316200
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 13nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-alpha serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316197
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-(3-aminoprop...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 16nM
Assay Description:
Inhibition of AKT
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-beta serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316184
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((S)-3-amino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 16nM
Assay Description:
Inhibition of AKT2
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
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PubMed
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Target
RAC-beta serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316194
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-6-((me...)
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Affinity Data
IC50: 16nM
Assay Description:
Inhibition of AKT2
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
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PubMed
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Target
RAC-beta serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316182
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((S)-2-amino...)
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Copy InChI
Affinity Data
Ki: 17nM
Assay Description:
Inhibition of AKT2
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-gamma serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316190
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((R)-2-amino...)
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Copy InChI
Affinity Data
IC50: 17nM
Assay Description:
Inhibition of AKT3
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-beta serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316191
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 20nM
Assay Description:
Inhibition of AKT2
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-beta serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316190
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((R)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 20nM
Assay Description:
Inhibition of AKT2
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-beta serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316201
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((S)-2-amino...)
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Affinity Data
IC50: 20nM
Assay Description:
Inhibition of AKT2
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-gamma serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316188
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-6-(pyr...)
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Affinity Data
IC50: 22nM
Assay Description:
Inhibition of AKT3
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-beta serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316193
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-(2-aminoethy...)
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Copy InChI
Affinity Data
IC50: 25nM
Assay Description:
Inhibition of AKT2
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-beta serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316192
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((R)-2-amino...)
Copy SMILES
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Affinity Data
IC50: 25nM
Assay Description:
Inhibition of AKT2
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-beta serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316182
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 25nM
Assay Description:
Inhibition of AKT2
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-beta serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316195
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-((dimethylam...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 25nM
Assay Description:
Inhibition of AKT2
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-gamma serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316187
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-(3-aminoprop...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 30nM
Assay Description:
Inhibition of AKT3
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
Target
RAC-beta serine/threonine-protein kinase
(Human)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50316189
(4-(2-(4-amino-1,2,5-oxadiazol-3-yl)-6-(2-aminoetho...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 39nM
Assay Description:
Inhibition of AKT2
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Date in BDB:
11/19/2010
Entry Details
Article
Copy BDB DOI
PubMed
Copy reaction URL
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