Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50028215
TargetIntegrin alpha-V(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50235980(2-((2S,5R,8S,11S)-5-benzyl-11-(3-guanidinopropyl)-...)
Affinity DataIC50:  0.130nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta5 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetIntegrin alpha-V(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50276748(CHEMBL460012 | [(1R,3S,9S,11S,14R)-9-(3-Guanidino-...)
Affinity DataIC50:  0.900nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta5 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50276748(CHEMBL460012 | [(1R,3S,9S,11S,14R)-9-(3-Guanidino-...)
Affinity DataIC50:  5.64nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta3 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50276746(CHEMBL452724 | c[RGDf-(3S)-Carboxymorpholine])
Affinity DataIC50:  15.1nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta5 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50235980(2-((2S,5R,8S,11S)-5-benzyl-11-(3-guanidinopropyl)-...)
Affinity DataIC50:  18.9nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta3 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetIntegrin alpha-V(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50276747(CHEMBL443362 | c[RGDf-(3R)-Carboxymorpholine])
Affinity DataIC50:  21nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta5 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50276747(CHEMBL443362 | c[RGDf-(3R)-Carboxymorpholine])
Affinity DataIC50:  32.6nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta3 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50276746(CHEMBL452724 | c[RGDf-(3S)-Carboxymorpholine])
Affinity DataIC50:  157nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta3 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed