Compile Data Set for Download or QSAR
maximum 50k data
Found 81 Enz. Inhib. hit(s) with all data for entry = 50028288
TargetHistamine H2 receptor(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50257636(5-(5-iodo-2-isopropyl-4-methoxyphenoxy)pyrimidine-...)
Affinity DataKi:  1.00E+8nMAssay Description:Inhibition of histamine H2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50257636(5-(5-iodo-2-isopropyl-4-methoxyphenoxy)pyrimidine-...)
Affinity DataKi:  1.00E+8nMAssay Description:Inhibition of 5HT6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50257636(5-(5-iodo-2-isopropyl-4-methoxyphenoxy)pyrimidine-...)
Affinity DataKi:  1.00E+8nMAssay Description:Inhibition of 5HT3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50257636(5-(5-iodo-2-isopropyl-4-methoxyphenoxy)pyrimidine-...)
Affinity DataKi:  1.00E+8nMAssay Description:Inhibition of 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413370(CHEMBL495204)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50257636(5-(5-iodo-2-isopropyl-4-methoxyphenoxy)pyrimidine-...)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413370(CHEMBL495204)
Affinity DataIC50:  13nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413395(CHEMBL495203)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413382(CHEMBL494833)
Affinity DataIC50:  25nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413394(CHEMBL448525)
Affinity DataIC50:  25nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413377(CHEMBL494176)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413400(CHEMBL521983)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413373(CHEMBL502618)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413395(CHEMBL495203)
Affinity DataIC50:  79nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50257636(5-(5-iodo-2-isopropyl-4-methoxyphenoxy)pyrimidine-...)
Affinity DataIC50:  79nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413378(CHEMBL523043)
Affinity DataIC50:  79nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413374(CHEMBL446310)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413397(CHEMBL492967)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413394(CHEMBL448525)
Affinity DataIC50:  100nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413403(CHEMBL521820)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413391(CHEMBL494772)
Affinity DataIC50:  126nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413373(CHEMBL502618)
Affinity DataIC50:  158nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413380(CHEMBL444469)
Affinity DataIC50:  158nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413398(CHEMBL500550)
Affinity DataIC50:  158nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413399(CHEMBL492968)
Affinity DataIC50:  158nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413383(CHEMBL494832)
Affinity DataIC50:  158nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413378(CHEMBL523043)
Affinity DataIC50:  316nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413398(CHEMBL500550)
Affinity DataIC50:  316nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413400(CHEMBL521983)
Affinity DataIC50:  316nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413374(CHEMBL446310)
Affinity DataIC50:  398nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413380(CHEMBL444469)
Affinity DataIC50:  398nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413377(CHEMBL494176)
Affinity DataIC50:  398nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413379(CHEMBL504607 | TCMDC-132471)
Affinity DataIC50:  398nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413372(CHEMBL494181)
Affinity DataIC50:  501nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413382(CHEMBL494833)
Affinity DataIC50:  501nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413399(CHEMBL492968)
Affinity DataIC50:  631nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413396(CHEMBL492562)
Affinity DataIC50:  631nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413397(CHEMBL492967)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413371(CHEMBL495195)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413390(CHEMBL494239)
Affinity DataIC50:  1.26E+3nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413369(CHEMBL494940)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413379(CHEMBL504607 | TCMDC-132471)
Affinity DataIC50:  1.59E+3nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413403(CHEMBL521820)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413393(CHEMBL494761)
Affinity DataIC50:  1.59E+3nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413381(CHEMBL494834)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413372(CHEMBL494181)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413391(CHEMBL494772)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413383(CHEMBL494832)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413396(CHEMBL492562)
Affinity DataIC50:  2.51E+3nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50413371(CHEMBL495195)
Affinity DataIC50:  2.51E+3nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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